SCHEMBL4538972

SCHEMBL4538972

N#Cc1ccc(S(=O)(=O)N2CCCCC2CNC(=O)C23CC4CC(CC(C4)C2)C3)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.46
CYP19A1 P11511 1/20 0.38
TRPV4 Q9HBA0 14/20 0.38
CYP3A4 P08684 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8063549 0.91 HSD11B1 (0.38) HSD11B1
SCHEMBL4537224 0.88 P2RX7 (0.43)
SCHEMBL8069525 0.87 EPHX2 (0.45) HSD11B1
SCHEMBL4530293 0.86 P2RX7 (0.44)
SCHEMBL4531364 0.85 HSD11B1 (0.44) HSD11B1
SCHEMBL4538974 0.84 CYP19A1 (0.39) HSD11B1CYP19A1TRPV4
SCHEMBL4537337 0.83 ATM (0.46) HSD11B1
SCHEMBL4542459 0.82 P2RX7 (0.42) HSD11B1
SCHEMBL4534371 0.80 DRD2 (0.41)
SCHEMBL4542906 0.80 TP53 (0.43) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed