SCHEMBL4539279

SCHEMBL4539279

O=[N+]([O-])c1c[nH]nc1C1CCOCC1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.38
TXNRD1 Q16881 2/20 0.38
PKM P14618 1/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
DAO P14920 1/20 0.34
BCL6 P41182 2/20 0.33
BCOR Q6W2J9 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CFTR P13569 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28899995 0.90 TXNRD1 (0.34) MAPTTXNRD1PKMCYP1A2CYP2C9
SCHEMBL2554448 0.89 GPR35 (0.33) MAPTTXNRD1CYP1A2ALDH1A1CYP2C19
SCHEMBL22572956 0.86 ALDH1A1 (0.34) MAPTTXNRD1ALDH1A1LMNAGAA
SCHEMBL22572955 0.84 MAPT (0.33) MAPTTXNRD1PKM
SCHEMBL22090173 0.81 TXNRD1 (0.36) MAPTTXNRD1ALDH1A1GAA
SCHEMBL22089936 0.79 JAK2 (0.34) TXNRD1ALDH1A1LMNA
SCHEMBL3786184 0.77 DAO (0.33) DAOCFTR
SCHEMBL23012286 0.75 DAO (0.33) DAO
SCHEMBL15556927 0.75 OPRL1 (0.33) DAO
SCHEMBL1559055 0.75 IRAK4 (0.33) DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638031-A1 PYRAZOLE AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2013-09-18 EP disclosed
WO-2012062783-A1 PYRAZOLE AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed