SCHEMBL4540574

SCHEMBL4540574

CCNc1ccnc(NC(C)=O)c1C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
KDM4E B2RXH2 2/20 0.40
HSD17B10 Q99714 1/20 0.40
PGK1 P00558 1/20 0.38
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
MAPK8 P45983 3/20 0.36
PIK3C3 Q8NEB9 3/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
PARP1 P09874 1/20 0.34
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
HTT P42858 1/20 0.33
GFER P55789 1/20 0.33
PLEC Q15149 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4540577 0.89 PGK1 (0.44) ALDH1A1HPGDKDM4EHSD17B10PGK1
SCHEMBL3569660 0.73 KDM4E (0.43) ALDH1A1HPGDKDM4EHSD17B10PGK1
SCHEMBL18992945 0.70 MKNK1 (0.40) ALDH1A1HPGDKDM4EHSD17B10MKNK1
SCHEMBL2904340 0.68 UTS2R (0.41) ALDH1A1HPGDKDM4EHSD17B10PGK1
SCHEMBL13964874 0.67 MME (0.48) ALDH1A1HPGDKDM4EHSD17B10MAPK8
SCHEMBL5264765 0.66 ALDH1A1 (0.41) ALDH1A1HPGDKDM4EHSD17B10MKNK1
SCHEMBL9512487 0.66 ALDH1A1 (0.45) ALDH1A1HPGDKDM4EHSD17B10MKNK1
SCHEMBL8600507 0.65 MKNK1 (0.41) ALDH1A1HPGDKDM4EHSD17B10MKNK1
SCHEMBL19310488 0.65 NOS2 (0.47) ALDH1A1HPGDKDM4EHSD17B10MAPK8
SCHEMBL5263528 0.65 PLK1 (0.45) ALDH1A1MKNK1MKNK2MAPK8GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140164-A1 6-AMINONICOTINAMIDE DERIVATIVES AS POTENT AND SELECTIVE HISTONE DEACETYLASE INHIBITORS CHIPSCREEN BIOSCIENCES LTD. (CN) 2009-11-19 WO disclosed