SCHEMBL5264765

SCHEMBL5264765

CCNc1cccc(C)c1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
MAPT P10636 6/20 0.41
HSD17B10 Q99714 2/20 0.41
POLB P06746 1/20 0.40
HPGD P15428 3/20 0.40
CYP3A4 P08684 2/20 0.40
MAPK1 P28482 1/20 0.40
TSHR P16473 1/20 0.40
RECQL P46063 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
TP53 P04637 1/20 0.39
BLM P54132 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
HTT P42858 3/20 0.38
GAA P10253 2/20 0.38
KDM4E B2RXH2 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1903512 0.84 KDM4E (0.50) ALDH1A1MAPTPOLBHPGDCYP3A4
SCHEMBL9512487 0.83 ALDH1A1 (0.45) ALDH1A1MAPTHSD17B10HPGDMAPK1
SCHEMBL5263528 0.81 PLK1 (0.45) ALDH1A1NPC1RAB9AMKNK1MKNK2
SCHEMBL14454097 0.80 POLB (0.43) ALDH1A1MAPTHSD17B10POLBHPGD
SCHEMBL16696027 0.80 P2RX7 (0.43) ALDH1A1MAPTHSD17B10POLBHPGD
SCHEMBL5261951 0.79 CA12 (0.47) ALDH1A1MAPTHSD17B10POLBTSHR
SCHEMBL3014819 0.77 PTGS2 (0.51) ALDH1A1MAPTPOLBHPGDCYP3A4
SCHEMBL311565 0.77 PARP1 (0.46) ALDH1A1MAPTHSD17B10POLBHPGD
SCHEMBL29623796 0.76 KDM4E (0.47) ALDH1A1HSD17B10POLBHPGDCYP3A4
SCHEMBL688886 0.75 GPR35 (0.62) ALDH1A1MAPTHPGDCYP3A4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740551-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105760-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed