SCHEMBL4542926

SCHEMBL4542926

COc1ccc(S(=O)(=O)N2CCCC2CNC(=O)[C]2CCCCCCC2)c(OC)c1.[CH2].[CH2]

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.54
NPC1 O15118 1/20 0.51
PAX8 Q06710 1/20 0.47
HCRTR1 O43613 1/20 0.44
HCRTR2 O43614 1/20 0.44
DRD2 P14416 2/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
SLC6A4 P31645 1/20 0.43
DRD3 P35462 1/20 0.43
HTR2B P41595 1/20 0.43
KCNH2 Q12809 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537171 0.97 RAB9A (0.51) RAB9ANPC1PAX8
SCHEMBL4536863 0.88 HCRTR1 (0.52) RAB9ANPC1PAX8HCRTR1HCRTR2
SCHEMBL4537598 0.85 ALDH1A1 (0.52) NPC1
SCHEMBL4538118 0.85 RAB9A (0.49) RAB9ANPC1PAX8HCRTR1HCRTR2
SCHEMBL4542922 0.84 RAB9A (0.49) RAB9ANPC1PAX8HCRTR1HCRTR2
SCHEMBL4541160 0.83 CYP19A1 (0.51) NPC1
SCHEMBL4542327 0.82 DRD2 (0.50) RAB9ADRD2
SCHEMBL4541692 0.82 RAB9A (0.47) RAB9ANPC1DRD2DRD3HTR2B
SCHEMBL4539820 0.81 RAB9A (0.67) RAB9ANPC1PAX8HCRTR1HCRTR2
SCHEMBL4537168 0.81 RAB9A (0.47) RAB9ANPC1PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed