SCHEMBL454919

SCHEMBL454919

Cc1[c]c(C2CC2)ccc1-c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.35
PDK2 Q15119 1/20 0.33
PDK4 Q16654 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
CYP2A6 P11509 1/20 0.33
CYP2B6 P20813 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PARP10 Q53GL7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL459103 0.80 ALDH1A1 (0.36) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL456741 0.80 KDM4E (0.31) KDM4EMEN1ALDH1A1MAPTHPGD
SCHEMBL457353 0.80 PDE4D (0.33) CYP2A6CYP2B6ALDH1A1MAPTNPSR1
SCHEMBL4371389 0.74 ESR2 (0.41) ESR2CYP2A6CYP2B6ALDH1A1HPGD
SCHEMBL15063871 0.71
SCHEMBL456995 0.71 ALDH1A1 (0.41) ESR2CYP2A6CYP2B6KDM4EALDH1A1
SCHEMBL456233 0.71 ESR2 (0.38) ESR2CYP2A6CYP2B6ALDH1A1HPGD
SCHEMBL6206554 0.71 CYP2A6 (0.41) ESR2CYP2A6CYP2B6KDM4EALDH1A1
SCHEMBL27714313 0.71 ESR2 (0.47) ESR2CYP2A6CYP2B6KDM4EMEN1
SCHEMBL28926395 0.69 BACE1 (0.44) ESR2CYP2A6CYP2B6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed