SCHEMBL457353

SCHEMBL457353

COc1[c]c(C2CC2)ccc1-c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.33
SLC6A3 Q01959 1/20 0.32
BACE1 P56817 1/20 0.31
SQOR Q9Y6N5 1/20 0.31
HRH1 P35367 1/20 0.31
DHODH Q02127 1/20 0.31
PDE4B Q07343 3/20 0.30
PDE4A P27815 1/20 0.30
PDE4C Q08493 1/20 0.30
CYP1A1 P04798 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2E1 P05181 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C8 P10632 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2A6 P11509 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP4B1 P13584 1/20 0.30
CYP2B6 P20813 1/20 0.30
CYP3A5 P20815 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL454919 0.80 ESR2 (0.35) HRH1CYP2A6CYP2B6ALDH1A1MAPT
SCHEMBL456741 0.75 KDM4E (0.31) HRH1ALDH1A1MAPTNPSR1
SCHEMBL7820403 0.74 PDE4B (0.38) PDE4DBACE1SQORPDE4BPDE4A
SCHEMBL456629 0.74 SQOR (0.39) PDE4DBACE1SQORPDE4BPDE4A
SCHEMBL458401 0.73 SQOR (0.34) PDE4DBACE1SQORPDE4BPDE4A
SCHEMBL455612 0.73 ALDH1A1 (0.38) PDE4DBACE1SQORPDE4BPDE4A
SCHEMBL457574 0.73 SQOR (0.38) PDE4DBACE1SQORPDE4BPDE4A
SCHEMBL21331773 0.71 BACE1 (0.42) PDE4DBACE1SQORPDE4BPDE4A
SCHEMBL456986 0.71 PDE4B (0.33) PDE4DSLC6A3BACE1SQORHRH1
SCHEMBL457181 0.68 ADRB2 (0.33) PDE4DBACE1SQORPDE4BPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed