SCHEMBL459103

SCHEMBL459103

Brc1[c]c(C2CC2)ccc1-c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
MAPK1 P28482 2/20 0.36
ANPEP P15144 2/20 0.33
IL1RN P18510 1/20 0.33
ERAP2 Q6P179 1/20 0.33
ERAP1 Q9NZ08 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HSD17B10 Q99714 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL454919 0.80 ESR2 (0.35) ALDH1A1CHRM2CHRM4CHRM5CHRM1
SCHEMBL456741 0.79 KDM4E (0.31) ALDH1A1ANPEPKDM4EMEN1MAPT
SCHEMBL457353 0.75 PDE4D (0.33) ALDH1A1MAPTNPSR1HRH1
SCHEMBL457364 0.72 ALDH1A1 (0.44) ALDH1A1MAPK1MAPTHPGDHSD17B10
SCHEMBL454901 0.69 ALDH1A1 (0.41) ALDH1A1MAPK1MAPTHPGDHSD17B10
SCHEMBL457524 0.69 ALDH1A1 (0.41) ALDH1A1MAPK1KDM4EHPGDNPSR1
SCHEMBL457102 0.66 ALDH1A1 (0.38) ALDH1A1MAPK1
SCHEMBL455777 0.64 RAB9A (0.41) ALDH1A1MAPK1MEN1KMT2ANPSR1
SCHEMBL16752251 0.64 AKR1C3 (0.31)
SCHEMBL16393627 0.62 BRD4 (0.51) ALDH1A1MAPK1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed