SCHEMBL4551501

SCHEMBL4551501

NC(=O)c1ccc(C(N)=O)n1S(=O)(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 2/20 0.46
CXCL8 P10145 1/20 0.44
NOD1 Q9Y239 1/20 0.44
CYP2D6 P10635 2/20 0.41
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
CYP2C9 P11712 2/20 0.40
CYP3A4 P08684 2/20 0.40
TSHR P16473 2/20 0.40
CYP2C19 P33261 2/20 0.40
MMP2 P08253 1/20 0.40
PKM P14618 1/20 0.40
PARL Q9H300 1/20 0.40
POLB P06746 1/20 0.40
PARP1 P09874 1/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836440 0.79 ALDH1A1 (0.62) SRCCXCL8NOD1MAPTALDH1A1
SCHEMBL5500240 0.73 CA12 (0.51) SRCNOD1MAPTALDH1A1LMNA
SCHEMBL3837213 0.73 PPARG (0.61) NOD1MAPTALDH1A1LMNA
SCHEMBL27700600 0.73 ALDH1A1 (0.53) SRCCXCL8NOD1MAPTALDH1A1
SCHEMBL31579035 0.73 HTR6 (0.52) SRCNOD1MAPTALDH1A1LMNA
SCHEMBL9789169 0.72 PKM (0.46) SRCALDH1A1LMNACYP3A4TSHR
SCHEMBL6911498 0.68 CYP2D6 (0.40) SRCCYP2D6ALDH1A1CYP2C9CYP3A4
(Phenylsulfonyl)Benzene SCHEMBL8958296 0.68 HTR6 (0.74) ALDH1A1LMNATSHRMMP2L3MBTL1
(Phenylsulfonyl)Benzene SCHEMBL28297601 0.68 HTR6 (0.74) ALDH1A1LMNATSHRMMP2L3MBTL1
SCHEMBL23440300 0.67 HSD11B1 (0.41) CXCL8ALDH1A1TSHRPOLBRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076492-A2 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS Merck & Co., Inc. (US) 2009-07-08 EP claimed
WO-2008054605-A2 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS MERCK & CO., INC. (US) 2008-05-08 WO claimed