SCHEMBL4554402

SCHEMBL4554402

Cc1nn(C)c(-n2nc(C)c3ccccc32)c1/C=C/C=O.[KH]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 1/20 0.37
CYP2C9 P11712 3/20 0.36
HPGD P15428 2/20 0.36
CYP1A2 P05177 1/20 0.36
RAB9A P51151 4/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 3/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
CYP11B1 P15538 3/20 0.35
CYP11B2 P19099 3/20 0.35
GAA P10253 3/20 0.33
CYP19A1 P11511 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
MAPT P10636 1/20 0.33
LMNA P02545 1/20 0.33
ELANE P08246 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL963496 0.87 HTT (0.47) GLSCYP2C9HPGDCYP1A2RAB9A
SCHEMBL965896 0.82 ALDH1A1 (0.51) GLSHPGDRAB9ASMN1; SMN2NPC1
SCHEMBL965897 0.82 ALDH1A1 (0.51) GLSHPGDRAB9ASMN1; SMN2NPC1
SCHEMBL4554904 0.80 RAB9A (0.34) CYP2C9HPGDCYP1A2RAB9ASMN1; SMN2
SCHEMBL964447 0.78 NPC1 (0.40) CYP2C9HPGDCYP1A2RAB9ASMN1; SMN2
SCHEMBL4553928 0.76 CA12 (0.35) CYP2C9HPGDCYP1A2RAB9ASMN1; SMN2
SCHEMBL963891 0.75 CYP1A2 (0.45) CYP2C9HPGDCYP1A2SMN1; SMN2ALDH1A1
SCHEMBL4554658 0.74 CYP1A2 (0.31) CYP2C9HPGDCYP1A2RAB9ASMN1; SMN2
SCHEMBL964450 0.74 NPC1 (0.36) GLSRAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL964449 0.74 NPC1 (0.36) GLSRAB9ASMN1; SMN2NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118066-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA Takeda Pharmaceutical Company Limited (JP) 2009-11-18 EP disclosed
WO-2008099794-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-08-21 WO disclosed