SCHEMBL4554658

SCHEMBL4554658

Cc1nn(C)c(-n2ccc3c(C)cccc32)c1/C=C/C=O.[KH]

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 1/20 0.31
FABP4 P15090 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554766 0.88 NOTUM (0.36) CYP1A2CYP2C9CYP2C19NPC1ALDH1A1
SCHEMBL963202 0.88 CYP1A2 (0.38) CYP1A2CYP2C9CYP2C19FABP4NPC1
SCHEMBL962156 0.84 ALDH1A1 (0.48) FABP4NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL962154 0.84 ALDH1A1 (0.48) FABP4NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL4553928 0.83 CA12 (0.35) CYP1A2CYP2C9CYP2C19NPC1ALDH1A1
SCHEMBL967577 0.76 CYP1A2 (0.42) CYP1A2CYP2C9CYP2C19ALDH1A1SMN1; SMN2
SCHEMBL4554436 0.75 MAPT (0.42)
SCHEMBL4554187 0.75 HTR2A (0.33) HTR2AHTR2C
SCHEMBL4554908 0.74 CDC7 (0.37) HTR2AHTR2C
SCHEMBL4553594 0.74 KDM4E (0.35) ALDH1A1HTR2AHTR2CHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118066-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA Takeda Pharmaceutical Company Limited (JP) 2009-11-18 EP disclosed
WO-2008099794-A1 FUSED RING COMPOUNDS AS PARTIAL AGONISTS OF PPAR-GAMMA TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-08-21 WO disclosed