SCHEMBL4559442

SCHEMBL4559442

CC(C)C(C#N)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.46
ESR1 P03372 4/20 0.44
ESR2 Q92731 4/20 0.44
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
CYP17A1 P05093 2/20 0.39
TRPA1 O75762 1/20 0.38
TSHR P16473 1/20 0.38
ACP3 P15309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL955278 0.87 TRPA1 (0.48) ESR1ESR2TRPA1TSHR
Hydrochloric Acid SCHEMBL5299628 0.85 TRPA1 (0.46) ESR1ESR2TRPA1TSHR
SCHEMBL954845 0.79 PTGS2 (0.48) PTGS2CTSSCTSKCHRNB2CHRNA4
SCHEMBL17455465 0.77 TSHR (0.48) PTGS2ESR1ESR2CHRNB2CHRNA4
SCHEMBL11878426 0.76 PTGS2 (0.46) PTGS2ESR1ESR2CTSSCTSK
SCHEMBL12019807 0.75 ALOX5AP (0.39) ESR1ESR2
SCHEMBL1193245 0.75 CHRNB2 (0.42) PTGS2ESR1ESR2CTSSCTSK
SCHEMBL10952365 0.75 ESR1 (0.47) ESR1ESR2CTSSCTSK
SCHEMBL10706998 0.75 ESR1 (0.75) ESR1ESR2
SCHEMBL7939324 0.75 ESR1 (0.47) ESR1ESR2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118496274-A Fluorine-containing probe for distinguishing and detecting chiral analytes, preparation and application thereof 中国科学院上海有机化学研究所 2024-08-16 CN disclosed
US-9771394-B2 Antimicrobial polymyxins for treatment of bacterial infections MICURX PHARMACEUTICALS, INC. (KY) 2017-09-26 US disclosed
US-9771394-B2 Antimicrobial polymyxins for treatment of bacterial infections MICURX PHARMACEUTICALS, INC. (KY) 2017-09-26 US disclosed
US-20160185823-A1 ANTIMICROBIAL POLYMYXINS FOR TREATMENT OF BACTERIAL INFECTIONS MICURX PHARMACEUTICALS, INC. 2016-06-30 US disclosed
US-20090291988-A1 Reversible Inhibitors of Monoamine Oxidase A and B MERCK FROSST CANADA LTD. (CA) 2009-11-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090291988-A1 Reversible Inhibitors of Monoamine Oxidase A and B MAOB, MAOA, XDH PTGS2 1499/4885ESR1 1417/4885ESR2 1622/4885
US-20160185823-A1 ANTIMICROBIAL POLYMYXINS FOR TREATMENT OF BACTERIAL INFECTIONS VIP, AQP1, PEF1 PTGS2 2904/4885ESR1 4584/4885ESR2 4693/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.