SCHEMBL4559535

SCHEMBL4559535

CC(C)=Cc1cc(N)ccc1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.38
THRB P10828 3/20 0.36
TDP1 Q9NUW8 3/20 0.36
RECQL P46063 2/20 0.36
POLB P06746 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
APEX1 P27695 1/20 0.36
BLM P54132 1/20 0.36
KMT2A Q03164 1/20 0.36
MCL1 Q07820 1/20 0.36
TSHR P16473 3/20 0.35
PDE10A Q9Y233 1/20 0.35
CYP3A4 P08684 5/20 0.35
ALDH1A1 P00352 3/20 0.35
ALOX15 P16050 3/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6312425 0.98 POLB (0.39) CASP1THRBTDP1RECQLPOLB
SCHEMBL19636018 0.81 CASP1 (0.48) CASP1THRBTDP1RECQLPOLB
SCHEMBL6311762 0.76 ALDH1A1 (0.33) THRBTDP1RECQLCYP3A4ALDH1A1
SCHEMBL6952023 0.75 GRIN2D (0.33) CASP1TDP1POLBMAPTTSHR
SCHEMBL24521736 0.75 NOS2 (0.33) CASP1USP2TSHRPDE10AALDH1A1
SCHEMBL5253253 0.74 CASP1 (0.40) CASP1THRBTDP1RECQLPOLB
SCHEMBL27523981 0.73 CYP3A4 (0.41) CASP1TDP1MEN1USP2MAPT
SCHEMBL29090092 0.71 CASP1 (0.39) CASP1THRBTDP1RECQLPOLB
SCHEMBL454407 0.71 CASP1 (0.39) CASP1THRBTDP1RECQLPOLB
SCHEMBL454405 0.71 CASP1 (0.39) CASP1THRBTDP1RECQLPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849766-B2 1,4-diamino-2-alkenylbenzene derivatives, and dyes containing these compounds WELLA AKTIENGESELLSCHAFT (DE) 2005-02-01 US claimed
EP-1351921-B1 NOVEL 1,4-DIAMINO-2-ALKENYL-BENZENE DERIVATIVES AND COLORANTS CONTAINING SAID COMPOUNDS WELLA AG (DE) 2004-12-01 EP claimed
US-20030121110-A1 Novel 1,4-diamino-2-alkenylbenzene derivatives , and dyes containing these compounds HFC PRESTIGE INTERNATIONAL OPERATIONS SWITZERLAND SÀRL (CH) 2003-07-03 US claimed
US-20090156441-A1 Cycloalkyl phenylenediamines as deposit control agents for lubricants GREAT LAKES CHEMICAL GLOBAL, INC. 2009-06-18 US disclosed
US-6849766-B2 1,4-diamino-2-alkenylbenzene derivatives, and dyes containing these compounds WELLA AKTIENGESELLSCHAFT (DE) 2005-02-01 US disclosed
EP-1351921-B1 NOVEL 1,4-DIAMINO-2-ALKENYL-BENZENE DERIVATIVES AND COLORANTS CONTAINING SAID COMPOUNDS WELLA AG (DE) 2004-12-01 EP disclosed
US-20030121110-A1 Novel 1,4-diamino-2-alkenylbenzene derivatives , and dyes containing these compounds HFC PRESTIGE INTERNATIONAL OPERATIONS SWITZERLAND SÀRL (CH) 2003-07-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030121110-A1 Novel 1,4-diamino-2-alkenylbenzene derivatives , and dyes containing these compounds AOC1, AOX1, GPX1 CASP1 550/4885THRB 3258/4885TDP1 261/4885
US-20090156441-A1 Cycloalkyl phenylenediamines as deposit control agents for lubricants C5, C9, C1S CASP1 3529/4885THRB 4816/4885TDP1 1337/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.