SCHEMBL456986

SCHEMBL456986

COc1[c]c(C2CC2)c(-c2ccccc2)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.33
PDE4D Q08499 4/20 0.33
PDE4A P27815 3/20 0.33
PDE4C Q08493 3/20 0.33
SLC6A3 Q01959 1/20 0.32
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
BACE1 P56817 1/20 0.31
SQOR Q9Y6N5 1/20 0.31
HRH1 P35367 1/20 0.31
DHODH Q02127 1/20 0.31
AKR1C3 P42330 1/20 0.30
AKR1C1 Q04828 1/20 0.30
CYP1A1 P04798 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2E1 P05181 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C8 P10632 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7820403 0.74 PDE4B (0.38) PDE4BPDE4DPDE4APDE4CALOX5AP
SCHEMBL2850552 0.67 IKBKB (0.43) PDE4BPDE4DPDE4APDE4CBACE1
SCHEMBL28039230 0.66 PDE4B (0.50) PDE4BPDE4DPDE4APDE4CALOX5AP
SCHEMBL454919 0.66 ESR2 (0.35) HRH1CYP2A6CYP2B6ALDH1A1MAPT
SCHEMBL15352348 0.65 ABCB1 (0.32)
SCHEMBL6130375 0.64 CTSD (0.42) BACE1ALDH1A1MAPTHTT
SCHEMBL2011554 0.63 CYP1A1 (0.50) DHODHCYP1A1CYP1A2CYP2E1CYP3A4
SCHEMBL1069430 0.63 ALDH1A1 (0.43) PDE4BPDE4DPDE4APDE4CCYP1A1
SCHEMBL336435 0.62 PDE4B (0.38) PDE4BPDE4DPDE4APDE4CCYP1A1
SCHEMBL458401 0.62 SQOR (0.34) PDE4BPDE4DPDE4APDE4CALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed