SCHEMBL457221

SCHEMBL457221

CCc1nc(-c2ccccc2)[c][nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.42
TP53 P04637 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ADORA3 P0DMS8 3/20 0.40
ADORA2A P29274 3/20 0.40
ADORA1 P30542 3/20 0.40
DDAH1 O94760 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
RAB9A P51151 3/20 0.35
ALDH1A1 P00352 3/20 0.34
MAPT P10636 2/20 0.34
DHFR P00374 1/20 0.34
HEXA P06865 1/20 0.34
HEXB P07686 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NPC1 O15118 2/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17599658 0.78 HEXA (0.41) RAB9AHEXAHEXBKDM4ENPC1
SCHEMBL7469061 0.75 KDM4E (0.41) SMN1; SMN2L3MBTL1ADORA3ADORA2AADORA1
SCHEMBL2097244 0.72 DCUN1D1 (0.41) SMN1; SMN2TNKS2NR1H2NR1H3RAB9A
SCHEMBL6497018 0.68 ALDH1A1 (0.50) SMN1; SMN2TP53ADORA3RAB9AALDH1A1
SCHEMBL457222 0.64 SMN1; SMN2 (0.56) SMN1; SMN2TP53L3MBTL1ADORA3ADORA2A
SCHEMBL1696584 0.64 NR1H2 (0.66) SMN1; SMN2TP53ADORA2ANR1H2NR1H3
SCHEMBL1696508 0.63 TP53 (0.53) SMN1; SMN2TP53L3MBTL1ADORA3ADORA2A
SCHEMBL458788 0.63 BTK (0.36) SMN1; SMN2TP53L3MBTL1ADORA3ADORA2A
SCHEMBL5378775 0.63 KDM4E (0.59) SMN1; SMN2TP53L3MBTL1ALDH1A1MAPT
SCHEMBL19116734 0.63 L3MBTL1 (0.61) SMN1; SMN2TP53L3MBTL1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed