SCHEMBL4572967

SCHEMBL4572967

COc1nc(N2CCN(C(=O)O)C(C)C2)ncc1C1CC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 5/20 0.46
PIK3CD O00329 10/20 0.41
PIK3R1 P27986 1/20 0.41
HCRTR2 O43614 3/20 0.41
GRM1 Q13255 1/20 0.39
CHRM2 P08172 2/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573572 0.86 GPR119 (0.51) CHRM4PIK3CDPIK3R1HCRTR2
SCHEMBL8108991 0.86 GPR119 (0.51) CHRM4PIK3CDPIK3R1HCRTR2
SCHEMBL4573090 0.84 CHRM4 (0.45) CHRM4PIK3CDPIK3R1HCRTR2GRM1
SCHEMBL4573074 0.83 CTSB (0.45) CHRM4GRM1
SCHEMBL4573353 0.78 CTSB (0.42) GRM1
SCHEMBL4573182 0.78 PIK3CD (0.41) CHRM4PIK3CDPIK3R1GRM1
SCHEMBL8113211 0.75 ROCK2 (0.39)
SCHEMBL21551483 0.74 GRM1 (0.48) CHRM4PIK3CDPIK3R1GRM1CHRM2
SCHEMBL4573206 0.73 PIK3CD (0.38) CHRM4PIK3CDPIK3R1GRM1
SCHEMBL18145739 0.73 CHRM1 (0.53) CHRM4PIK3CDPIK3R1GRM1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed