SCHEMBL4573909

SCHEMBL4573909

COc1cnc(C2CC2)c(N2CCN(C(=O)OC(C)(C)C)C(C)C2)n1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.46
GPR119 Q8TDV5 2/20 0.44
SUV39H2 Q9H5I1 2/20 0.43
HDAC1 Q13547 1/20 0.43
IDH1 O75874 6/20 0.36
NR1H2 P55055 2/20 0.36
NR1H3 Q13133 2/20 0.36
GRM1 Q13255 1/20 0.36
PIK3CD O00329 2/20 0.35
SETD7 Q8WTS6 1/20 0.35
PDE10A Q9Y233 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8108577 1.00 MAP4K4 (0.46) MAP4K4GPR119SUV39H2HDAC1IDH1
SCHEMBL4573206 0.86 PIK3CD (0.38) IDH1GRM1PIK3CD
SCHEMBL8116228 0.86 MAP4K4 (0.48) MAP4K4GPR119SUV39H2HDAC1NR1H2
SCHEMBL4584298 0.86 MAP4K4 (0.48) MAP4K4GPR119SUV39H2HDAC1NR1H2
SCHEMBL4573072 0.82 MAP4K4 (0.51) MAP4K4GPR119SUV39H2HDAC1GRM1
SCHEMBL4573109 0.82 MAP4K4 (0.51) MAP4K4GPR119SUV39H2HDAC1GRM1
SCHEMBL8113244 0.78 MAP4K4 (0.52) MAP4K4GPR119SUV39H2HDAC1NR1H2
SCHEMBL4584408 0.78 MAP4K4 (0.52) MAP4K4GPR119SUV39H2HDAC1NR1H2
SCHEMBL8108991 0.76 GPR119 (0.51) MAP4K4GPR119SUV39H2HDAC1PIK3CD
SCHEMBL4573572 0.76 GPR119 (0.51) MAP4K4GPR119SUV39H2HDAC1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed