SCHEMBL457803

SCHEMBL457803

CCCc1[c]c(F)c(-c2ccccc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
HPGD P15428 3/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
MAPT P10636 2/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
ADRB2 P07550 1/20 0.31
NPC1 O15118 1/20 0.31
PKM P14618 1/20 0.31
RAB9A P51151 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SOAT1 P35610 1/20 0.31
PTGS1 P23219 3/20 0.30
MEN1 O00255 2/20 0.30
PTGS2 P35354 2/20 0.30
KMT2A Q03164 2/20 0.30
FABP2 P12104 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457978 0.86 TP53 (0.32) ADORA3ADORA2AADORA1HPGDMAPT
SCHEMBL458760 0.81 ESR2 (0.34) ADORA3ADORA2AADORA1HPGDSMN1; SMN2
SCHEMBL457181 0.80 ADRB2 (0.33) ADORA3ADORA2AADORA1MAPTALDH1A1
SCHEMBL456773 0.79 CYP2A6 (0.35) ADORA3ADORA2AADORA1HPGDSMN1; SMN2
SCHEMBL457437 0.79 ADORA3 (0.33) ADORA3ADORA2AADORA1HPGDSMN1; SMN2
SCHEMBL14675940 0.72 ESR2 (0.38) HPGDMAPTALDH1A1HSD17B10PTGS1
SCHEMBL10428951 0.71 BACE1 (0.36) HPGDMAPTALDH1A1HSD17B10PTGS1
SCHEMBL4155256 0.71 PSMB5 (0.38) SOAT1TSHRPSMB5
SCHEMBL456919 0.68 ALDH1A1 (0.41) ADORA1HPGDMAPTALDH1A1HSD17B10
SCHEMBL7814278 0.68 CYP2A6 (0.41) HPGDMAPTALDH1A1HSD17B10PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed