SCHEMBL458760

SCHEMBL458760

CCCc1[c]c(C)c(-c2ccccc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
PSMB5 P28074 1/20 0.33
CYP2A6 P11509 1/20 0.32
CYP2B6 P20813 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
HSD11B1 P28845 2/20 0.32
MAPT P10636 2/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
ADRB2 P07550 1/20 0.32
NPC1 O15118 1/20 0.32
PKM P14618 1/20 0.32
RAB9A P51151 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457803 0.81 ADORA3 (0.33) ESR2ADORA3ADORA2AADORA1PSMB5
SCHEMBL457437 0.81 ADORA3 (0.33) ADORA3ADORA2AADORA1PSMB5SMN1; SMN2
SCHEMBL456773 0.81 CYP2A6 (0.35) ESR2ADORA3ADORA2AADORA1PSMB5
SCHEMBL457181 0.78 ADRB2 (0.33) ADORA3ADORA2AADORA1MAPTALDH1A1
SCHEMBL4371389 0.72 ESR2 (0.41) ESR2PDCD1CD274PSMB5CYP2A6
SCHEMBL4155256 0.72 PSMB5 (0.38) PSMB5HSD11B1TSHRGCGR
SCHEMBL6206554 0.69 CYP2A6 (0.41) ESR2PDCD1CD274CYP2A6CYP2B6
SCHEMBL456995 0.69 ALDH1A1 (0.41) ESR2PDCD1CD274CYP2A6CYP2B6
SCHEMBL456233 0.69 ESR2 (0.38) ESR2ADORA3ADORA2AADORA1PDCD1
SCHEMBL456470 0.68 TP53 (0.34) ESR2ADORA3ADORA2AADORA1PDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed