SCHEMBL4589967

SCHEMBL4589967

C=CCC(OC(N)=O)C(C)(C)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.44
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
ALDH1A1 P00352 3/20 0.40
CYP2C19 P33261 2/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.36
KDM4E B2RXH2 1/20 0.36
HIF1A Q16665 1/20 0.36
KIF11 P52732 1/20 0.35
GAA P10253 1/20 0.35
CYP2D6 P10635 3/20 0.34
CYP1A2 P05177 2/20 0.34
EPHX1 P07099 3/20 0.34
MEN1 O00255 1/20 0.34
PKM P14618 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAPK1 P28482 1/20 0.33
LMNA P02545 1/20 0.33
CHRM2 P08172 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4589971 0.82 ALDH1A1 (0.37) HTTKMT2AMAPTALDH1A1CYP2C19
SCHEMBL9049034 0.82 MAPT (0.44) HTTKMT2AMAPTCYP2C19SMN1; SMN2
SCHEMBL28939289 0.76 LMNA (0.33) MAPTTSHRLMNACHRM2CHRM1
SCHEMBL22115533 0.75 MAPT (0.33) KMT2AMAPTCYP2C19KIF11CYP1A2
SCHEMBL4375323 0.74 CYP2C19 (0.49) HTTKMT2AMAPTALDH1A1CYP2C19
SCHEMBL2969422 0.73 MAPT (0.48) KMT2AMAPTALDH1A1CYP2C19TSHR
SCHEMBL4588810 0.72 CYP2C19 (0.47) HTTALDH1A1CYP2C19SMN1; SMN2CYP2D6
SCHEMBL18426754 0.71 CYP2C19 (0.53) CYP2C19SMN1; SMN2CYP2D6CYP1A2PKM
SCHEMBL28738770 0.69 MAPT (0.47) HTTKMT2AMAPTALDH1A1CYP2C19
SCHEMBL11005490 0.69 HTT (0.55) HTTKMT2AMAPTALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937656-A1 7-(2-AMINO-1-HYDROXY-ETHYL)-4-HYDROXYBENZOTHIAZOL-2(3H)-ONE-DERIVATIVES AS BETA 2 ADRENOCEPTOR AGONISTS AstraZeneca AB (SE) 2008-07-02 EP disclosed
WO-2007027134-A1 7-(2-AMINO-1-HYDROXY-ETHYL)-4-HYDROXYBENZOTHIAZOL-2(3H)-ONE-DERIVATIVES AS β2 ADRENOCEPTOR AGONISTS ASTRAZENECA AB (SE) 2007-03-08 WO disclosed