SCHEMBL4593434

SCHEMBL4593434

ClC(Cl)(C1(c2ccccc2)N=NN=N1)C1(c2ccccc2)N=NN=N1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.35
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
TAAR1 Q96RJ0 1/20 0.32
P2RX1 P51575 1/20 0.32
P2RX3 P56373 1/20 0.32
P2RX4 Q99571 1/20 0.32
P2RX7 Q99572 1/20 0.32
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5280778 0.86 TSHR (0.35) TSHRMAOAMAOB
SCHEMBL5277316 0.82 TSHR (0.32) TSHR
SCHEMBL4592879 0.78 ACHE (0.38) TAAR1
SCHEMBL4594159 0.77 ACHE (0.35) TSHRMAOAMAOB
SCHEMBL4593190 0.77 SLC6A3 (0.33) MAOAMAOB
SCHEMBL5277372 0.76 OPRM1 (0.35)
SCHEMBL5275595 0.76 MAOB (0.39) TSHRMAOAMAOB
SCHEMBL2008502 0.76 KDM1A (0.45) TSHRTAAR1
SCHEMBL9205048 0.74 KCNN4 (0.33) TSHR
SCHEMBL4593785 0.74 TSHR (0.35) TSHRTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP disclosed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO disclosed