SCHEMBL4593785

SCHEMBL4593785

Clc1ccccc1C1(C(Cl)(Cl)C2(c3ccccc3Cl)N=NN=N2)N=NN=N1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
LMNA P02545 1/20 0.35
TAAR1 Q96RJ0 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
PDK2 Q15119 2/20 0.33
GRIN1 Q05586 2/20 0.32
GRIN2A Q12879 2/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
HDAC4 P56524 1/20 0.32
PNMT P11086 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593846 0.78 HTR2A (0.33) PDK2
SCHEMBL4593251 0.78 TSHR (0.33) TSHRPDK2HDAC4
SCHEMBL4593434 0.74 TSHR (0.35) TSHRTAAR1
SCHEMBL4593447 0.71 DRD1 (0.32)
SCHEMBL5280778 0.66 TSHR (0.35) TSHR
SCHEMBL4594159 0.63 ACHE (0.35) TSHRLMNAIDO1
SCHEMBL5277316 0.63 TSHR (0.32) TSHR
SCHEMBL4593190 0.63 SLC6A3 (0.33) IDO1
SCHEMBL4593654 0.60 MAOA (0.40) TSHRTAAR1IDO1
SCHEMBL31506444 0.60 LMNA (0.45) TSHRLMNATAAR1CRHBPCRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP disclosed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO disclosed