SCHEMBL4593869

SCHEMBL4593869

COC(=O)C(Cc1cc(C)c2[nH]nnc2c1)NC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.38
TACR3 P29371 1/20 0.38
PARP1 P09874 1/20 0.38
PARP3 Q9Y6F1 1/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
ALDH1A1 P00352 1/20 0.38
THRB P10828 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
PYGL P06737 1/20 0.37
POLB P06746 1/20 0.37
NLRP3 Q96P20 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3587642 1.00 ATM (0.38) ATMTACR3PARP1PARP3CYP2C9
SCHEMBL13030993 0.86 ALDH1A1 (0.49) ALDH1A1CYP3A4
SCHEMBL13030997 0.83 ALDH1A1 (0.38) ALDH1A1THRB
Hydrochloric Acid SCHEMBL3551035 0.82 ALDH1A1 (0.40) ALDH1A1THRB
Hydrochloric Acid SCHEMBL3551031 0.82 ALDH1A1 (0.40) ALDH1A1THRB
SCHEMBL3547969 0.78 MMP8 (0.38) ATMALDH1A1HSD17B10POLB
SCHEMBL3761588 0.76 L3MBTL1 (0.37) ATMPARP1PARP3ALDH1A1HSD17B10
SCHEMBL3608214 0.76 PKM (0.43) CYP2C9ALDH1A1THRBHSD17B10CYP3A4
SCHEMBL3761591 0.74 TRPM8 (0.36) ATMTACR3PARP1PARP3CYP2C9
SCHEMBL4586241 0.72 LNPEP (0.45) ATMCYP2C9CYP2C19ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689493-A4 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2008-04-23 EP disclosed
EP-1689493-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS Bristol-Myers Squibb Pharma Company (US) 2006-08-16 EP disclosed
WO-2005065779-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-21 WO disclosed