SCHEMBL4598027

SCHEMBL4598027

O=C1NC[C@](c2cccc(F)c2)(C2CCOCC2)N1C1CCNCC1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
SLC6A2 P23975 1/20 0.32
CHRNB4 P30926 1/20 0.32
SLC6A4 P31645 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC6A3 Q01959 1/20 0.32
HTR6 P50406 5/20 0.32
KDM1A O60341 2/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
OPRM1 P35372 2/20 0.31
OPRL1 P41146 2/20 0.31
BACE1 P56817 1/20 0.31
PLAT P00750 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM3 P20309 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596506 0.87 DRD2 (0.34) CHRNA1CHRNB1CHRNB2SLC6A2CHRNB4
SCHEMBL4596625 0.87 HTR2C (0.35) CHRNA1CHRNB1CHRNB2SLC6A2CHRNB4
SCHEMBL4597256 0.87 DRD2 (0.34) CHRNA1CHRNB1CHRNB2SLC6A2CHRNB4
SCHEMBL4596041 0.87 KDM4E (0.32) KDM1AKDM4EALDH1A1OPRM1OPRL1
SCHEMBL4597510 0.87 KDM4E (0.32) KDM1AKDM4EALDH1A1OPRM1OPRL1
SCHEMBL4596707 0.78 GABRA1 (0.32)
SCHEMBL4597792 0.77 CHRM2 (0.34) SLC6A2SLC6A4SLC6A3BACE1PLAT
SCHEMBL4625414 0.77 CHRM2 (0.34) SLC6A2SLC6A4SLC6A3BACE1PLAT
SCHEMBL4596366 0.77 CHRM2 (0.37) SLC6A4SLC6A3HTR6OPRM1OPRL1
SCHEMBL4596721 0.77 CHRM2 (0.37) SLC6A4SLC6A3HTR6OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed