SCHEMBL4597825

SCHEMBL4597825

O=C1NCC(c2ccc(F)cc2)(c2cccc(Cl)c2)N1C1CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.39
CHRM3 P20309 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
SLC6A9 P48067 1/20 0.37
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
TACR1 P25103 1/20 0.35
CHRM1 P11229 2/20 0.35
DRD2 P14416 2/20 0.34
NPY5R Q15761 1/20 0.34
MAPK14 Q16539 2/20 0.34
KCNH2 Q12809 1/20 0.34
DPP4 P27487 1/20 0.34
DPP9 Q86TI2 1/20 0.34
HTR6 P50406 3/20 0.33
FADS1 O60427 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598352 0.84 SLC6A4 (0.41) DRD2KCNH2DPP4DPP9HTR6
SCHEMBL5179386 0.80 GRIN1 (0.38) CHRM2CHRM3HTR2AHTR2CHTR6
SCHEMBL4596721 0.76 CHRM2 (0.37) CHRM2CHRM3CYP2D6CYP2C9CYP2C19
SCHEMBL4596366 0.76 CHRM2 (0.37) CHRM2CHRM3CYP2D6CYP2C9CYP2C19
SCHEMBL4597529 0.76 BACE1 (0.38) CYP2D6CYP2C9CYP2C19HTR2AHTR2C
SCHEMBL4597256 0.73 DRD2 (0.34) CYP2D6CYP2C9CYP2C19HTR2AHTR2C
SCHEMBL4596506 0.73 DRD2 (0.34) CYP2D6CYP2C9CYP2C19HTR2AHTR2C
SCHEMBL4597871 0.72 SLC6A2 (0.40) DRD2KCNH2DPP4DPP9HTR6
SCHEMBL4597579 0.72 DRD2 (0.33) CYP2D6CYP2C9CYP2C19HTR2AHTR2C
SCHEMBL4598182 0.71 GRIN1 (0.36) CHRM2CHRM3CYP2C19TP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed