SCHEMBL4597256

SCHEMBL4597256

O=C1NC[C@](c2cccc(Cl)c2)(C2CCOCC2)N1C1CCNCC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
DPP4 P27487 3/20 0.33
DPP9 Q86TI2 2/20 0.33
BACE1 P56817 2/20 0.33
HTR6 P50406 3/20 0.33
SLC6A4 P31645 2/20 0.33
CYP2C19 P33261 2/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
ADRB1 P08588 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTR1A P08908 1/20 0.33
CYP2D6 P10635 1/20 0.33
THRB P10828 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596506 1.00 DRD2 (0.34) DRD2GABRA1GABRG2GABRB3DPP4
SCHEMBL4596721 0.90 CHRM2 (0.37) DRD2GABRA1GABRG2GABRB3DPP4
SCHEMBL4596366 0.90 CHRM2 (0.37) DRD2GABRA1GABRG2GABRB3DPP4
SCHEMBL4598027 0.87 CHRNA1 (0.32) BACE1HTR6SLC6A4CHRNA1CHRNB1
SCHEMBL4596625 0.87 HTR2C (0.35) BACE1ADRB1HTR2AHTR2CHTR2B
SCHEMBL4597510 0.87 KDM4E (0.32) BACE1MEN1ALDH1A1KMT2A
SCHEMBL4596041 0.87 KDM4E (0.32) BACE1MEN1ALDH1A1KMT2A
SCHEMBL4597579 0.85 DRD2 (0.33) DRD2GABRA1GABRG2GABRB3DPP4
SCHEMBL4596707 0.78 GABRA1 (0.32) GABRA1GABRG2GABRB3
SCHEMBL4597792 0.75 CHRM2 (0.34) BACE1SLC6A4TP53HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed