SCHEMBL4596698

SCHEMBL4596698

CN(C(=O)O)C1Cc2cccc(-c3ccc(Cl)cc3Cl)c2O1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 1/20 0.39
EDNRA P25101 1/20 0.39
AQP1 P29972 2/20 0.38
HTR1A P08908 2/20 0.37
HTR7 P34969 2/20 0.37
KIF11 P52732 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 3/20 0.36
POLB P06746 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSP90AA1 P07900 1/20 0.35
NPSR1 Q6W5P4 3/20 0.35
HTT P42858 3/20 0.35
LMNA P02545 2/20 0.35
S1PR2 O95136 1/20 0.35
S1PR4 O95977 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595391 0.88 HTR1A (0.41) HTR1AHTR7KIF11ALDH1A1MAPT
SCHEMBL4595383 0.86 HTR7 (0.43) EDNRBEDNRAHTR1AHTR7ALDH1A1
SCHEMBL6047972 0.85 AQP1 (0.42) AQP1KIF11ALDH1A1MAPTPOLB
SCHEMBL4595037 0.85 HTR7 (0.45) HTR1AHTR7KIF11
SCHEMBL15758703 0.83 MAPT (0.34) HTR1AHTR7ALDH1A1MAPTNPC1
SCHEMBL15759012 0.81 TDP1 (0.39) HTR1AHTR7ALDH1A1POLBHPGD
SCHEMBL4596574 0.80 ALDH1A1 (0.40) EDNRBEDNRAHTR7KIF11ALDH1A1
SCHEMBL4225937 0.79 HTR7 (0.43) HTR1AHTR7ALDH1A1POLBMEN1
SCHEMBL4596973 0.79 HTR1A (0.41) HTR1AHTR7KIF11ALDH1A1POLB
SCHEMBL4596752 0.77 RAB9A (0.38) EDNRBEDNRAHTR1AHTR7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
WO-2007030150-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH (US) 2007-03-15 WO disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed