SCHEMBL4600429

SCHEMBL4600429

O=Cc1c(Cl)c(-c2ccccc2)cc(Cl)c1OC(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
THRA P10827 2/20 0.34
THRB P10828 2/20 0.34
ACLY P53396 2/20 0.33
RAB9A P51151 1/20 0.33
METAP2 P50579 1/20 0.33
FFAR4 Q5NUL3 2/20 0.33
AR P10275 1/20 0.33
FFAR1 O14842 1/20 0.33
CYP2C9 P11712 1/20 0.33
SCN5A Q14524 1/20 0.33
CYP2A6 P11509 1/20 0.33
SLC22A12 Q96S37 3/20 0.32
KDM4E B2RXH2 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HSP90AA1 P07900 1/20 0.32
CHRM5 P08912 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29213635 0.74 MEN1 (0.42) MEN1KMT2AALDH1A1TDP1ACLY
SCHEMBL4600326 0.73 AR (0.35) MEN1KMT2ARAB9AMETAP2FFAR4
SCHEMBL10973832 0.72 ALDH1A1 (0.45) MEN1KMT2AALDH1A1THRBACLY
SCHEMBL4276345 0.70 ALDH1A1 (0.42) MEN1KMT2AALDH1A1THRBACLY
SCHEMBL6535943 0.69 ALDH1A1 (0.45) MEN1KMT2AALDH1A1THRBRAB9A
SCHEMBL30583087 0.69 CYP2A6 (0.50) THRATHRBMETAP2FFAR4CYP2A6
SCHEMBL27907871 0.69 CYP2A6 (0.50) THRATHRBMETAP2FFAR4CYP2A6
SCHEMBL4032566 0.69 LMNA (0.38) MEN1KMT2AALDH1A1TDP1THRB
SCHEMBL6535972 0.69 FFAR4 (0.43) MEN1KMT2AALDH1A1RAB9AFFAR4
SCHEMBL2041747 0.69 MEN1 (0.35) MEN1KMT2AALDH1A1TDP1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910292-A1 PIPERIDINE DERIVATIVE AS TACHYKININ RECEPTOR ANTAGONIST Takeda Pharmaceutical Company Limited (JP) 2008-04-16 EP disclosed
WO-2007015588-A1 PIPERIDINE DERIVATIVE AS TACHYKININ RECEPTOR ANTAGONIST TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-08 WO disclosed