SCHEMBL4603740

SCHEMBL4603740

C#CCOc1c(F)cc(C(=O)N(C)C2CCCCC2C)cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
TAS1R2 Q8TE23 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
S1PR3 Q99500 2/20 0.33
KMT2A Q03164 2/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PDK2 Q15119 4/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
POLB P06746 1/20 0.31
MAPK14 Q16539 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4603967 0.79 MAOA (0.34) MAOAMAOB
SCHEMBL4246193 0.77 TAS1R3 (0.58) TAS1R3TAS1R1TAS1R2
SCHEMBL4246190 0.77 TAS1R3 (0.58) TAS1R3TAS1R1TAS1R2
SCHEMBL4247030 0.77 TAS1R3 (0.58) TAS1R3TAS1R1TAS1R2
SCHEMBL4603140 0.77 MAOB (0.43) TAS1R3TAS1R1SIGMAR1TSHRMAOB
SCHEMBL2282332 0.77 TAS1R3 (0.41) TAS1R3TAS1R1TAS1R2MAPK14
SCHEMBL4242303 0.76 TAS1R3 (0.42) TAS1R3TAS1R1TAS1R2MAPK14
SCHEMBL4246293 0.76 TDP1 (0.39) TAS1R3TAS1R1TAS1R2TDP1KMT2A
SCHEMBL4242205 0.75 TAS1R3 (0.55) TAS1R3TAS1R1TAS1R2
SCHEMBL4602859 0.74 RIPK1 (0.33) MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940780-A1 AMIDE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL CO., LTD. (JP) 2008-07-09 EP disclosed
WO-2007049728-A1 AMIDE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-05-03 WO disclosed