SCHEMBL4604120

SCHEMBL4604120

O=C(O)c1ccc(-c2ccccc2)cc1NC(=O)C1CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 10/20 0.58
HDAC3 O15379 1/20 0.58
HDAC1 Q13547 1/20 0.58
HDAC2 Q92769 1/20 0.58
GSK3B P49841 2/20 0.54
PIK3CD O00329 1/20 0.54
PIM1 P11309 1/20 0.54
PIK3CA P42336 1/20 0.54
PIK3CG P48736 1/20 0.54
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 1/20 0.52
ADORA3 P0DMS8 1/20 0.51
ADORA2A P29274 1/20 0.51
ADORA1 P30542 1/20 0.51
GRIK1 P39086 1/20 0.50
PTPN1 P18031 1/20 0.50
HNF4A P41235 1/20 0.50
ACMSD Q8TDX5 1/20 0.50
GSK3A P49840 1/20 0.50
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2270149 0.93 ACLY (0.57) ACLYHDAC3HDAC1HDAC2KDM4E
SCHEMBL4617520 0.86 PRSS12 (0.56) ACLYHDAC3HDAC1HDAC2KDM4E
SCHEMBL3918325 0.85 HDAC1 (0.64) ACLYHDAC3HDAC1HDAC2KDM4E
SCHEMBL28170369 0.82 ALDH1A1 (0.60) HDAC3HDAC1HDAC2KDM4EALDH1A1
SCHEMBL16404476 0.82 ALDH1A1 (0.60) HDAC3HDAC1HDAC2KDM4EALDH1A1
SCHEMBL11727165 0.81 ACLY (0.62) ACLYHDAC3HDAC1HDAC2GRIK1
SCHEMBL4602392 0.81 HDAC1 (0.56) ACLYHDAC3HDAC1HDAC2KDM4E
SCHEMBL4604141 0.80 DHODH (0.48) ACLYHDAC3HDAC1HDAC2KDM4E
SCHEMBL2276115 0.80 MEN1 (0.49) ACLYKDM4EALDH1A1
SCHEMBL2270696 0.80 GAA (0.60) KDM4EALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940786-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C Arrow Therapeutics Limited (GB) 2008-07-09 EP disclosed
WO-2007031791-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2007-03-22 WO disclosed