SCHEMBL4607479

SCHEMBL4607479

CC(O)C(Oc1cccc2[nH]c3ccccc3c12)N1CCN(C(=O)c2cnc3ccccc3n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.45
GRM5 P41594 1/20 0.39
ADRB3 P13945 9/20 0.38
ADRB2 P07550 9/20 0.38
ADRB1 P08588 8/20 0.38
DNM1 Q05193 1/20 0.37
LANCL2 Q9NS86 1/20 0.37
DPP4 P27487 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4608590 0.85 RAB9A (0.46) ADRB3ADRB2ADRB1
SCHEMBL2996791 0.81 ADRB2 (0.58) PTK2ADRB3ADRB2ADRB1DNM1
SCHEMBL4607629 0.79 KDM4E (0.52)
SCHEMBL4608607 0.79 ALDH1A1 (0.44) ADRB3ADRB2ADRB1
SCHEMBL4606968 0.78 ADRB3 (0.42) ADRB3ADRB2ADRB1DNM1
SCHEMBL4607733 0.78 POLB (0.40) ADRB3ADRB2ADRB1DNM1
SCHEMBL4605749 0.78 TLR9 (0.49) ADRB3ADRB2ADRB1
SCHEMBL4608603 0.76 ADRB3 (0.49) ADRB3ADRB2ADRB1
SCHEMBL4605132 0.75 ADRB3 (0.46) ADRB3ADRB2ADRB1DNM1
SCHEMBL4608251 0.75 MITF (0.43) ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP claimed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO claimed
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP disclosed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO disclosed