SCHEMBL4616588

SCHEMBL4616588

CC(CS(=O)(=O)O)c1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
ALDH1A1 P00352 1/20 0.43
TSHR P16473 2/20 0.42
LMNA P02545 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
KCNA5 P22460 5/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KCNH2 Q12809 1/20 0.40
KDM4E B2RXH2 3/20 0.39
SLC6A3 Q01959 2/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
CYP2C19 P33261 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP2D6 P10635 1/20 0.38
KCNE1 P15382 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31501528 1.00 CYP1A2 (0.44) CYP1A2CYP3A4ALDH1A1TSHRLMNA
SCHEMBL5760051 1.00 CYP1A2 (0.44) CYP1A2CYP3A4ALDH1A1TSHRLMNA
SCHEMBL17309424 0.84 TSHR (0.43) CYP1A2CYP3A4ALDH1A1TSHRLMNA
SCHEMBL18263710 0.82 SLC6A2 (0.46) CYP1A2CYP3A4ALDH1A1TSHRLMNA
SCHEMBL28225638 0.81 KDM4E (0.44) CYP1A2CYP3A4ALDH1A1TSHRLMNA
SCHEMBL16696883 0.78 SLC6A2 (0.50) CYP1A2CYP3A4ALDH1A1TSHRLMNA
SCHEMBL6052780 0.78 CYP1A2 (0.45) CYP1A2CYP3A4ALDH1A1TSHRLMNA
SCHEMBL4807002 0.77 CYP1A2 (0.47) CYP1A2CYP3A4ALDH1A1TSHRLMNA
SCHEMBL14928678 0.76 TSHR (0.48) CYP1A2CYP3A4ALDH1A1TSHRLMNA
SCHEMBL30211265 0.76 TSHR (0.48) CYP1A2CYP3A4ALDH1A1TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12421200-B2 Manganese-catalysed hydrogenation of esters UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS (GB) 2025-09-23 US disclosed
US-12281058-B2 Manganese catalysts and their use in hydrogenation of ketones UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS (GB) 2025-04-22 US disclosed
WO-2024100405-A1 CATALYTIC HYDROGENATION PROCESS UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS (GB) 2024-05-16 WO disclosed
EP-3737663-B1 MANGANESE-CATALYSED HYDROGENATION OF ESTERS UNIV COURT UNIV ST ANDREWS (GB) 2023-02-22 EP disclosed
US-20220119329-A1 Manganese Catalysts and Their Use in Hydrogenation of Ketones UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS (GB) 2022-04-21 US disclosed
EP-3908588-A1 MANGANESE CATALYSTS AND THEIR USE IN HYDROGENATION OF KETONES University Court of The University of St Andrews (GB) 2021-11-17 EP disclosed
US-20210053932-A1 MANGANESE-CATALYSED HYDROGENATION OF ESTERS UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS (GB) 2021-02-25 US disclosed
EP-3737663-A1 MANGANESE-CATALYSED HYDROGENATION OF ESTERS University Court of The University of St Andrews (GB) 2020-11-18 EP disclosed
WO-2020144476-A1 MANGANESE CATALYSTS AND THEIR USE IN HYDROGENATION OF KETONES UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS (GB) 2020-07-16 WO disclosed
EP-1748975-B1 METHOD FOR THE PRODUCTION OF OPTICALLY ACTIVE 3-ALKYL CARBOXYLIC ACIDS AND THE INTERMEDIATE PRODUCTS THEREOF WACKER CHEMIE AG (DE) 2008-02-13 EP disclosed
EP-1325003-B1 7-CHLORO-4-HYDROXY-2-(2-PYRIDYLETHYL)-1,2,5,10-TETRAHYDROPYRIDAZINO 4,5-B|QUINOLINE-1,10-DIONE AND THE USE THEREOF FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-08-02 EP disclosed
US-6933297-B2 7-chloro-4-hydroxy-2-(2-pyridylethyl)-1,2,5,10-tetrahydropyridazino[4,5-b]quinoline-1,10-dione and the use thereof for the treatment of pain ASTRAZENECA AB (CH) 2005-08-23 US disclosed
US-20040053930-A1 7-Chloro-4-hydroxy-2-(2-pyridylethyl)-1,2,5,10-tetrahydropyridazino[4,5-b]quinoline-1,10-dione and the use thereof for the treatment of pain ASTRAZENECA AB (SE) 2004-03-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040053930-A1 7-Chloro-4-hydroxy-2-(2-pyridylethyl)-1,2,5,10-tetrahydropyridazino[4,5-b]quinoline-1,10-dione and the use thereof for the treatment of pain HTR5A, OPRK1, OPRD1 CYP1A2 66/4885CYP3A4 40/4885ALDH1A1 179/4885
US-12281058-B2 Manganese catalysts and their use in hydrogenation of ketones CYC1, SCO2, MT-CO3 CYP1A2 1170/4885CYP3A4 1922/4885ALDH1A1 2055/4885
US-12421200-B2 Manganese-catalysed hydrogenation of esters ADH5, HDHD5, ADH1A CYP1A2 337/4885CYP3A4 93/4885ALDH1A1 1003/4885
US-20210053932-A1 MANGANESE-CATALYSED HYDROGENATION OF ESTERS ADH5, HDHD5, ADH1A CYP1A2 337/4885CYP3A4 93/4885ALDH1A1 1003/4885
US-20220119329-A1 Manganese Catalysts and Their Use in Hydrogenation of Ketones CYC1, SCO2, MT-CO3 CYP1A2 1170/4885CYP3A4 1922/4885ALDH1A1 2055/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.