SCHEMBL4622940

SCHEMBL4622940

CCCCCCOC(=O)[C@H](CCC(N)=O)NC(=O)c1ccc2c(c1)C(=O)c1ccccc1-2

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.44
ACHE P22303 2/20 0.44
CACNA1F O60840 1/20 0.44
CACNA1D Q01668 1/20 0.44
CACNA1S Q13698 1/20 0.44
CACNA1C Q13936 1/20 0.44
MAPK14 Q16539 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ATM Q13315 1/20 0.42
NOD1 Q9Y239 1/20 0.41
TAS1R3 Q7RTX0 3/20 0.40
TAS1R1 Q7RTX1 3/20 0.40
PTPRC P08575 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
MCHR1 Q99705 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2246525 0.91 NPC1 (0.43) MAPK14NPC1RAB9AATMPTPRC
SCHEMBL4621148 0.82 MAPT (0.55) MAPK14NPC1RAB9AATMPTPRC
SCHEMBL2249427 0.80 CA2 (0.59) MAPK14NPC1RAB9AATMPTPRC
SCHEMBL2248134 0.79 POLB (0.52) MAPK14NPC1RAB9AATMPTPRC
SCHEMBL4623235 0.79 RAB9A (0.43) ACHEMAPK14NPC1RAB9AATM
SCHEMBL2244945 0.79 PTPRC (0.47) MAPK14NPC1RAB9AATMPTPRC
SCHEMBL3587576 0.76 CCKBR (0.51)
SCHEMBL10425308 0.75 ALDH1A1 (0.56) NPC1RAB9A
SCHEMBL7350261 0.75 NOD1 (0.49) BCHEACHECACNA1FCACNA1DCACNA1S
SCHEMBL8430970 0.75 NOD1 (0.49) BCHEACHECACNA1FCACNA1DCACNA1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902014-A2 GLUTAMATE AGGRECANASE INHIBITORS Wyeth (US) 2008-03-26 EP claimed
WO-2007008994-A2 GLUTAMATE AGGRECANASE INHIBITORS WYETH (US) 2007-01-18 WO claimed