SCHEMBL4629167

SCHEMBL4629167

O=C(Cc1ccccc1)Nc1cccc(-c2ccccc2)c1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.57
HPGD P15428 3/20 0.57
LMNA P02545 4/20 0.57
KDM4E B2RXH2 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
KMT2A Q03164 5/20 0.54
MEN1 O00255 4/20 0.54
GAA P10253 3/20 0.54
L3MBTL1 Q9Y468 3/20 0.54
CASP3 P42574 1/20 0.53
SELL P14151 1/20 0.52
SELP P16109 1/20 0.52
SELE P16581 1/20 0.52
RAB9A P51151 1/20 0.51
PARP14 Q460N5 1/20 0.51
EPHX2 P34913 1/20 0.50
ATM Q13315 1/20 0.50
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
GPR35 Q9HC97 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4629164 0.77 ALDH1A1 (0.75) ALDH1A1HPGDLMNAKDM4ESMN1; SMN2
SCHEMBL12998051 0.77 ALDH1A1 (0.55) ALDH1A1HPGDLMNASMN1; SMN2KMT2A
SCHEMBL4803124 0.77 LMNA (0.58) ALDH1A1HPGDLMNAKDM4ESMN1; SMN2
SCHEMBL3393320 0.76 RAB9A (0.58) ALDH1A1HPGDLMNAKDM4ESMN1; SMN2
SCHEMBL11900441 0.76 ALDH1A1 (0.70) ALDH1A1HPGDLMNAKDM4ESMN1; SMN2
SCHEMBL4040223 0.74 ALDH1A1 (0.82) ALDH1A1HPGDLMNAKDM4ESMN1; SMN2
SCHEMBL4802411 0.73 LMNA (0.54) ALDH1A1HPGDLMNAKDM4ESMN1; SMN2
SCHEMBL8437112 0.73 ALDH1A1 (0.79) ALDH1A1HPGDLMNAKDM4ESMN1; SMN2
SCHEMBL6164465 0.73 LMNA (0.64) ALDH1A1HPGDLMNAKDM4ESMN1; SMN2
SCHEMBL593127 0.73 FOLH1 (0.61) ALDH1A1HPGDSMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633716-A4 BIARYLMETHYL INDOLINES, INDOLES AND TETRAHYDROQUINOLINES, USEFUL AS SERINE PROTEASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2008-03-26 EP claimed
EP-1633716-A2 BIARYLMETHYL INDOLINES, INDOLES AND TETRAHYDROQUINOLINES, USEFUL AS SERINE PROTEASE INHIBITORS Bristol-Myers Squibb Company (US) 2006-03-15 EP claimed
WO-2004094372-A2 COMPOUNDS USEFUL AS SERINE PROTEASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-04 WO claimed