SCHEMBL4629576

SCHEMBL4629576

CCc1cccc(CC)c1CN1C=NCC1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.40
GABRA1 P14867 3/20 0.34
GABRB2 P47870 3/20 0.34
HTR1A P08908 4/20 0.34
DRD2 P14416 3/20 0.33
DRD4 P21917 3/20 0.33
HTR2A P28223 3/20 0.33
HTR2C P28335 3/20 0.33
DRD3 P35462 3/20 0.33
KCNH2 Q12809 1/20 0.32
SCN5A Q14524 1/20 0.32
KMT2A Q03164 1/20 0.30
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9446985 0.79 COMT (0.37) KMT2A
SCHEMBL7118352 0.76 MPO (0.35)
SCHEMBL9447066 0.75 ADRA2B (0.38) HTR1AKMT2AADRA2AADRA2BADRA2C
SCHEMBL9447121 0.72 MAPT (0.51) HTR1ADRD2KMT2A
SCHEMBL9447022 0.70 HTR1A (0.46) HTR1AKCNH2KMT2AADRA2AADRA2B
SCHEMBL30537761 0.67 CYP19A1 (0.41) DRD4
SCHEMBL30332718 0.66 CYP19A1 (0.41) DRD4
SCHEMBL4099257 0.66 CYP2A13 (0.59) KMT2A
Hydrochloric Acid SCHEMBL28560184 0.65
SCHEMBL245773 0.64 GABRA1 (0.57) TAAR1GABRA1GABRB2HTR1AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed