SCHEMBL4630178

SCHEMBL4630178

CN1CCC(Nc2cccc(S(=O)(=O)c3cc4cc(Br)ccc4[nH]3)c2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.44
HRH4 Q9H3N8 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
CNR1 P21554 2/20 0.37
CYP3A4 P08684 2/20 0.36
ITK Q08881 1/20 0.36
BCAT1 P54687 1/20 0.35
CYP2D6 P10635 1/20 0.35
AXL P30530 1/20 0.35
VCP P55072 1/20 0.35
BRD4 O60885 3/20 0.35
JAK2 O60674 1/20 0.35
PDE5A O76074 1/20 0.35
ATAD2 Q6PL18 1/20 0.35
IDH2 P48735 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
HTR7 P34969 1/20 0.35
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630173 0.88 HRH4 (0.45) HTR6HRH4HRH3VCPHTR1A
SCHEMBL4629545 0.88 VCP (0.47) HTR6HRH4VCPHTR2A
SCHEMBL4630016 0.87 CA2 (0.46) HTR6HRH4HRH3CNR1BCAT1
Hydrochloric Acid SCHEMBL4628914 0.87 VCP (0.46) HTR6HRH4VCPHTR1AHTR2A
SCHEMBL4630008 0.85 HTR6 (0.42) HTR6HRH4HRH3CYP3A4ITK
SCHEMBL4628912 0.83 CYP3A4 (0.41) HRH4HRH3CNR1CYP3A4CYP2D6
SCHEMBL4629550 0.82 POLB (0.44) HTR6HRH4HRH3CNR1ITK
SCHEMBL4630007 0.81 CYP3A4 (0.49) HTR6HRH4HRH3CYP3A4CYP2D6
SCHEMBL4629706 0.79 HTR6 (0.45) HTR6HRH4CNR1AXLPDE5A
SCHEMBL2273734 0.75 HTR6 (0.54) HTR6CYP3A4HTR1ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919896-A1 AMINOARYL SULPHONAMIDE DERIVATIVES AS FUNCTIONAL 5-HT6 LIGANDS. Suven Life Sciences Limited (IN) 2008-05-14 EP disclosed
WO-2007020652-A1 AMINOARYL SULPHONAMIDE DERIVATIVES AS FUNCTIONAL 5-HT6 LIGANDS. SUVEN LIFE SCIENCES LIMITED (IN) 2007-02-22 WO disclosed