SCHEMBL463438

SCHEMBL463438

Cc1ccc(F)c([C@H]2CNC[C@@]2(NC(=O)OC(C)(C)C)c2ncc(OCCN3CCCCC3)cn2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
ESR1 P03372 3/20 0.35
ESR2 Q92731 3/20 0.35
ACHE P22303 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
PSMB1 P20618 1/20 0.33
PSMB5 P28074 1/20 0.33
PSMB2 P49721 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
AXL P30530 1/20 0.33
KDM4E B2RXH2 2/20 0.33
EPHX2 P34913 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
FLT3 P36888 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457491 0.79 ITGB3 (0.34)
SCHEMBL460033 0.78 RET (0.33)
SCHEMBL459944 0.76 NTRK1 (0.34)
SCHEMBL458010 0.76 ITGB3 (0.34)
SCHEMBL457723 0.76 NTRK1 (0.34) MEN1KMT2A
SCHEMBL457628 0.74 GPR119 (0.34)
SCHEMBL459071 0.74 NTRK1 (0.33) MEN1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL459362 0.71
SCHEMBL463286 0.70
SCHEMBL459500 0.69 HTT (0.34) MEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011147951-A1 CYCLOAMINO DERIVATIVES AS GPR119 ANTAGONISTS PROSIDION LIMITED (GB) 2011-12-01 WO disclosed