SCHEMBL4636714

SCHEMBL4636714

NCc1cccc(S(=O)(=O)C2CNCCO2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.37
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
SLC6A2 P23975 7/20 0.34
NCF1 P14598 1/20 0.33
HTR1A P08908 1/20 0.33
SLC6A4 P31645 6/20 0.32
PNMT P11086 1/20 0.31
ENPP2 Q13822 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31
SLC6A3 Q01959 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2897608 0.85 CA1 (0.42) CA12CA1CA2CA4CA6
SCHEMBL28153720 0.83 LMNA (0.44) DRD2DRD3HTR1ACA12CA1
SCHEMBL7671592 0.80 DRD2 (0.52) HTR6DRD2DRD3SLC6A2HTR1A
SCHEMBL6422590 0.79 SLC6A2 (0.38) HTR6DRD2DRD3SLC6A2HTR1A
SCHEMBL28092048 0.78 PKM (0.41)
SCHEMBL28285086 0.78 LMNA (0.42) DRD2DRD3
SCHEMBL28091851 0.77 AKR1C3 (0.47) CA1CA2
SCHEMBL7674336 0.77 HTR6 (0.47) HTR6SLC6A2SLC6A4SLC6A3
SCHEMBL14775611 0.74 HTR6 (0.37) HTR6SLC6A2SLC6A4CA12CA1
SCHEMBL28433779 0.74 HTR6 (0.39) HTR6CA12CA1CA2CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937652-B1 PYRIMIDINE AMIDE COMPOUNDS AS PGDS INHIBITORS AVENTIS PHARMA INC (US) 2014-07-30 EP disclosed
EP-1937652-A1 PYRIMIDINE AMIDE COMPOUNDS AS PGDS INHIBITORS Aventis Pharmaceuticals Inc. (US) 2008-07-02 EP disclosed
WO-2007041634-A1 PYRIMIDINE AMIDE COMPOUNDS AS PGDS INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2007-04-12 WO disclosed