SCHEMBL4637121

SCHEMBL4637121

FC(F)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
CHRNB2 P17787 1/20 0.50
CHRNA4 P43681 1/20 0.50
ACP3 P15309 2/20 0.46
PTGS2 P35354 1/20 0.46
KIF11 P52732 1/20 0.44
CYP3A4 P08684 2/20 0.43
MAPK1 P28482 1/20 0.43
CYP1A2 P05177 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MMP3 P08254 1/20 0.43
BCL2L1 Q07817 1/20 0.43
CYP17A1 P05093 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL60955 0.82
Hydrochloric Acid SCHEMBL28033934 0.79 DPP4 (0.45) ALDH1A1CYP3A4TAAR1TDP1
Hydrogen Sulfide SCHEMBL27610802 0.79 ALDH1A1 (0.60) ALDH1A1CHRNB2CHRNA4ACP3PTGS2
SCHEMBL16426382 0.79 PTGS2 (0.54) ALDH1A1CHRNB2CHRNA4ACP3PTGS2
SCHEMBL662302 0.78 PGK1 (0.38) KIF11
SCHEMBL1538543 0.77 RXRA (0.47) ALDH1A1CHRNB2CHRNA4PTGS2KIF11
SCHEMBL2838545 0.77 ALDH1A1 (0.56) ALDH1A1CHRNB2CHRNA4ACP3PTGS2
SCHEMBL13092431 0.76 CHRNA7 (0.42) ALDH1A1KIF11HSD17B10TDP1
SCHEMBL1539040 0.76 TSHR (0.43)
Biphenyl SCHEMBL6252617 0.76 ALDH1A1 (0.64) ALDH1A1CHRNB2CHRNA4PTGS2KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118932350-A Method for synthesizing carboxylic acid and deuterated carboxylic acid compound through electrochemical defluorination 江西师范大学 2024-11-12 CN disclosed
CN-117865773-A Preparation method of difluoromethyl aromatic compound based on palladium-catalyzed decarbonylation coupling 大连理工大学 2024-04-12 CN disclosed
EP-3053875-B1 FLUORINATING AGENT DAIKIN IND LTD (JP) 2022-09-28 EP disclosed
CN-110655539-B Method for synthesizing cis-difluoromethylcyclohexane derivatives and heterocyclic compounds by hydrogenation 四川大学 2021-11-12 CN disclosed
CN-111574322-A Preparation method of difluoromethyl aromatic compound 南京工业大学 2020-08-25 CN disclosed
WO-2020037109-A1 PROCESSES FOR FLUORINATION DOW AGROSCIENCES LLC (US) 2020-02-20 WO disclosed
CN-110655539-A Method for synthesizing cis-difluoromethylcyclohexane derivatives and heterocyclic compounds by hydrogenation 四川大学 2020-01-07 CN disclosed
US-10479681-B2 Fluorinating agent DAIKIN INDUSTRIES, LTD. (JP) 2019-11-19 US disclosed
US-20190152779-A1 FLUORINATING AGENT DAIKIN INDUSTRIES, LTD. (JP) 2019-05-23 US disclosed
US-10233080-B2 Fluorinating agent DAIKIN INDUSTRIES, LTD. (JP) 2019-03-19 US disclosed
US-9475756-B2 Difluoromethylation of aryl and vinyl iodides THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-10-25 US disclosed
US-9475756-B2 Difluoromethylation of aryl and vinyl iodides THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-10-25 US disclosed
US-9475756-B2 Difluoromethylation of aryl and vinyl iodides THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-10-25 US disclosed
EP-3053875-A1 FLUORINATING AGENT Daikin Industries, Ltd. (JP) 2016-08-10 EP disclosed
US-20150045580-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-02-12 US disclosed
US-20150045580-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-02-12 US disclosed
US-20150045580-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-02-12 US disclosed
WO-2013134296-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-09-12 WO disclosed
EP-1931425-A1 ANTITUBERCULOUS COMPOSITION COMPRISING OXAZOLE COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-06-18 EP disclosed
WO-2007043542-A1 ANTITUBERCULOUS COMPOSITION COMPRISING OXAZOLE COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-04-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10479681-B2 Fluorinating agent AFF2, AFF4, AFF1 ALDH1A1 2167/4885CHRNB2 3476/4885CHRNA4 3228/4885
US-10233080-B2 Fluorinating agent AFF2, AFF4, AFF1 ALDH1A1 2167/4885CHRNB2 3476/4885CHRNA4 3228/4885
US-20190152779-A1 FLUORINATING AGENT AFF2, AFF4, AFF1 ALDH1A1 2167/4885CHRNB2 3476/4885CHRNA4 3228/4885
US-20150045580-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES CUL2, CUL3, CYP4F2 ALDH1A1 2999/4885CHRNB2 2523/4885CHRNA4 3536/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.