SCHEMBL4638369

SCHEMBL4638369

CC(C)(C)C1c2ccc(N3CC[C@H](NC(=O)OCc4ccccc4)C3=O)c(F)c2CCCN1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
ACHE P22303 2/20 0.38
MGAT2 Q10469 1/20 0.37
CASP3 P42574 1/20 0.37
FKBP1A P62942 2/20 0.37
CASP1 P29466 2/20 0.36
FPR1 P21462 4/20 0.35
FPR2 P25090 4/20 0.35
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638371 0.86 CTSK (0.39) PARP1CA1CA2ACHECASP1
SCHEMBL4921278 0.80 TMEM97 (0.39) PARP1CA1CA2ACHECASP3
SCHEMBL5277552 0.79 CA1 (0.39) CA1CA2ACHECASP3FKBP1A
SCHEMBL5242559 0.73
SCHEMBL4638357 0.72 CTSL (0.43) CA1ACHECASP1CTSK
SCHEMBL149797 0.70 CASP3 (0.43) CA1CA2ACHECASP3CASP1
SCHEMBL4706101 0.68 ALDH1A1 (0.45) CASP3CASP1CTSK
SCHEMBL8302634 0.68 SRD5A1 (0.43) FPR1FPR2
SCHEMBL4858641 0.68 SRD5A1 (0.43) FPR1FPR2
SCHEMBL5241778 0.68 TDP1 (0.35) FPR1FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951712-A2 CHEMICAL COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-08-06 EP disclosed
WO-2007059952-A2 1-BENZAZEPINE-3-SULFONYLAMINO-2-PYRRLORIDONES AS FACTOR XA INHIBITORS GLAXO GROUP LIMITED (GB) 2007-05-31 WO disclosed