SCHEMBL4640097

SCHEMBL4640097

CC(C)(C)COC(=O)N[C@@H](Cn1cnc2c(N3CCC(C(=O)O)CC3)ncnc21)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
SIRT3 Q9NTG7 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
KMT2A Q03164 3/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 4/20 0.34
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
ITGB3 P05106 4/20 0.34
ITGAV P06756 4/20 0.34
HRH4 Q9H3N8 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MTOR P42345 1/20 0.33
HTR2C P28335 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6805959 0.92 ITGB3 (0.40) TDP1KMT2APOLBMAPTKDM4E
SCHEMBL27524220 0.89 ITGB3 (0.46) CNR1CNR2ITGB3ITGAVHRH4
SCHEMBL4640164 0.89 ITGB3 (0.46) CNR1CNR2ITGB3ITGAVHRH4
SCHEMBL6810270 0.87 NPEPPS (0.34) TDP1SIRT2SIRT1SIRT3CNR1
SCHEMBL27474218 0.84 KMT2A (0.39) TDP1SIRT2SIRT1SIRT3KMT2A
SCHEMBL4640715 0.84 KMT2A (0.39) TDP1SIRT2SIRT1SIRT3KMT2A
SCHEMBL4641013 0.84 ITGB3 (0.34) SIRT2SIRT1SIRT3KMT2AMAPT
SCHEMBL6884541 0.82 KMT2A (0.34) TDP1SIRT2SIRT1SIRT3CNR1
SCHEMBL27475141 0.82 KMT2A (0.34) TDP1SIRT2SIRT1SIRT3CNR1
SCHEMBL6805865 0.82 TDP1 (0.41) TDP1SIRT2SIRT1SIRT3CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853084-B1 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AG (DE) 2008-08-13 EP disclosed
US-6723727-B1 VITRONECTIN RECEPTOR ANTAGONISTS; INHIBITORS OF BONE RESORPTION; OSTEOPOROSIS HOECHST AKTIENGESELLSCHAFT (DE) 2004-04-20 US disclosed
EP-0853084-A2 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-07-15 EP disclosed