SCHEMBL4640355

SCHEMBL4640355

CCOC(=O)Oc1ccc2ncn(CCC(C)(C)N)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.49
MTNR1B P49286 1/20 0.49
CA2 P00918 1/20 0.45
F10 P00742 2/20 0.39
TNF P01375 2/20 0.39
POLB P06746 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
MEN1 O00255 1/20 0.37
F2 P00734 1/20 0.37
PRSS1 P07477 1/20 0.37
GAA P10253 2/20 0.36
HPGD P15428 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640769 0.92 CA2 (0.44) MTNR1AMTNR1BCA2F10TNF
SCHEMBL4641222 0.84 MTNR1A (0.45) MTNR1AMTNR1BCA2F10POLB
SCHEMBL4826368 0.83 ALDH1A1 (0.38) MTNR1AMTNR1BCA2F10TNF
SCHEMBL4916141 0.82 NPC1 (0.48) MTNR1AMTNR1BCA2F10TNF
SCHEMBL4775013 0.81 ALDH1A1 (0.38) MTNR1AMTNR1BCA2F10TNF
SCHEMBL4777107 0.78 TNF (0.36) CA2F10TNFALDH1A1MAPT
SCHEMBL4638928 0.77 TRPM5 (0.35) CA2F10TNFALDH1A1MAPT
SCHEMBL4893401 0.76 CNR2 (0.39) MTNR1AMTNR1BF10TNFPOLB
SCHEMBL4913399 0.76 NPC1 (0.47) F10MAPTSMN1; SMN2KMT2AMEN1
SCHEMBL4915876 0.75 CA1 (0.42) CA2TNFPOLBALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed