SCHEMBL4664156

SCHEMBL4664156

COc1cccc(CC2CCC(O)(c3ccc(Cl)c(C(F)(F)F)c3)C(C)(N(C)C)C2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.40
OPRM1 P35372 8/20 0.40
OPRD1 P41143 4/20 0.40
OPRK1 P41145 2/20 0.40
HTR1A P08908 2/20 0.40
SLC6A4 P31645 2/20 0.40
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR1D P28221 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR7 P34969 1/20 0.40
HRH1 P35367 1/20 0.40
DRD3 P35462 1/20 0.40
HTR2B P41595 1/20 0.40
HTR5A P47898 1/20 0.40
HTR6 P50406 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4664225 0.84 OPRL1 (0.49) GRIN2BOPRM1OPRD1OPRK1HTR1A
SCHEMBL4663525 0.80 OPRK1 (0.49) OPRM1OPRD1OPRK1SLC6A4SLC6A2
SCHEMBL4665572 0.73 OPRL1 (0.47) GRIN2BOPRM1OPRD1OPRK1HTR1A
SCHEMBL4665942 0.70 SMN1; SMN2 (0.38) OPRM1OPRD1OPRK1SLC6A4SLC6A2
SCHEMBL4665533 0.69 TRPA1 (0.38) OPRM1SLC6A4DRD2DRD4SLC6A2
SCHEMBL5170874 0.69 OPRM1 (0.39) GRIN2BOPRM1OPRD1OPRK1HTR1A
SCHEMBL5170803 0.68 OPRM1 (0.39) GRIN2BOPRM1OPRD1OPRK1HTR1A
SCHEMBL4663394 0.67 OPRK1 (0.53) OPRM1OPRD1OPRK1SLC6A4SLC6A2
SCHEMBL4665743 0.67 SLC6A4 (0.41) OPRM1OPRD1OPRK1HTR1ASLC6A4
SCHEMBL4663720 0.67 OPRK1 (0.60) OPRM1OPRD1OPRK1SLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1571140-B1 C-substituted cyclohexylmethylamine derivatives GRUENENTHAL GMBH (DE) 2008-11-12 EP claimed