SCHEMBL4665533

SCHEMBL4665533

CN(C)C1(C)CC(Cc2ccc(Cl)cc2)CCC1(O)c1ccc(Cl)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
SLC6A4 P31645 3/20 0.37
SLC6A3 Q01959 3/20 0.37
CCR5 P51681 1/20 0.36
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRL1 P41146 1/20 0.35
AVPR1A P37288 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CHIT1 Q13231 2/20 0.34
KCNH2 Q12809 1/20 0.34
SLC6A2 P23975 2/20 0.34
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4665942 0.88 SMN1; SMN2 (0.38) TRPA1SLC6A4SLC6A3CCR5OPRM1
SCHEMBL4665489 0.83 TRPA1 (0.38) TRPA1SLC6A4SLC6A3CCR5OPRM1
SCHEMBL4665552 0.78 STS (0.43) TRPA1CCR5ALDH1A1ATP1A1ATP1B1
SCHEMBL4665899 0.78 CXCR4 (0.36) TRPA1SLC6A4SLC6A3CCR5OPRM1
SCHEMBL4664225 0.78 OPRL1 (0.49) TRPA1SLC6A4SLC6A3DRD2DRD4
SCHEMBL29693296 0.74 ALDH1A1 (0.43) TRPA1CCR5ALDH1A1P2RX7
SCHEMBL4665379 0.70 OPRK1 (0.42) SLC6A4SLC6A3OPRM1ALDH1A1SLC6A2
SCHEMBL4665371 0.67 OPRK1 (0.39) SLC6A4SLC6A3CCR5OPRM1ALDH1A1
SCHEMBL4663483 0.66 DRD2 (0.41) TRPA1SLC6A4SLC6A3DRD2DRD4
SCHEMBL4664046 0.65 SMN1; SMN2 (0.48) SLC6A4OPRM1ALDH1A1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1571140-B1 C-substituted cyclohexylmethylamine derivatives GRUENENTHAL GMBH (DE) 2008-11-12 EP claimed