SCHEMBL4670084

SCHEMBL4670084

NC(=O)c1ccc(-n2nnn(Cc3ccccc3)c2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.56
MAPK1 P28482 1/20 0.54
ATM Q13315 1/20 0.54
PLA2G10 O15496 1/20 0.46
PLA2G2A P14555 1/20 0.46
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
HPGD P15428 3/20 0.45
HCAR3 P49019 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 2/20 0.43
TSHR P16473 1/20 0.43
GAA P10253 1/20 0.42
PARP10 Q53GL7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4673352 0.85 MAPK1 (0.50) ROCK2MAPK1ATMPLA2G10PLA2G2A
SCHEMBL4670186 0.84 EPHX2 (0.48) ROCK2MAPK1ATMCYP2C9CYP2C19
SCHEMBL4670086 0.83 ROCK2 (0.61) ROCK2CYP2C19HPGDTSHR
SCHEMBL4673552 0.79 MAPK1 (0.49) ROCK2MAPK1ATMHPGDMEN1
SCHEMBL4675102 0.78 ALDH1A1 (0.42) MAPK1ATMHPGDHCAR3MEN1
SCHEMBL4675660 0.76 ROCK2 (0.56) ROCK2MEN1KMT2AALDH1A1
SCHEMBL4670479 0.73 ALDH1A1 (0.39) MAPK1ATMHPGDMEN1KMT2A
SCHEMBL4672091 0.72 ALDH1A1 (0.47) MAPK1ATMHPGDMEN1KMT2A
SCHEMBL19643312 0.72 ROCK2 (1.00) ROCK2
SCHEMBL4670468 0.72 PARP15 (0.42) MAPK1ATMCYP2C9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054881-B1 NOVEL SULFONAMIDE SUBSTITUTED CHROMAN DERIVATIVES USEFUL AS BETA-3 ADRENORECEPTOR AGONISTS BAYER CORP (US) 2008-07-30 EP disclosed