SCHEMBL4675102

SCHEMBL4675102

CCCn1nnn(-c2ccc(C(N)=O)cc2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
MAPK1 P28482 1/20 0.41
ATM Q13315 1/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
HCAR3 P49019 1/20 0.41
TSHR P16473 1/20 0.40
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA10 Q9GZZ6 1/20 0.39
CHRNA9 Q9UGM1 1/20 0.39
KDM4E B2RXH2 2/20 0.39
POLB P06746 2/20 0.39
ALPL P05186 1/20 0.39
GAA P10253 1/20 0.39
ALPG P10696 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4670479 0.83 ALDH1A1 (0.39) ALDH1A1MAPK1ATMMEN1KMT2A
SCHEMBL4670427 0.82 ADORA2B (0.41) ALDH1A1ADORA2AADORA2BSMN1; SMN2
Hydrochloric Acid SCHEMBL9384727 0.81 ADORA2B (0.40) ALDH1A1ADORA2AADORA2BMEN1KMT2A
SCHEMBL4672091 0.80 ALDH1A1 (0.47) ALDH1A1MAPK1ATMMEN1KMT2A
SCHEMBL4673352 0.79 MAPK1 (0.50) ALDH1A1MAPK1ATMMEN1KMT2A
SCHEMBL4670468 0.79 PARP15 (0.42) ALDH1A1MAPK1ATMMEN1KMT2A
SCHEMBL4670421 0.79 PARP10 (0.42) ALDH1A1MAPK1ATMMEN1KMT2A
SCHEMBL4677832 0.78 PARP15 (0.43) MAPK1ATMMEN1KMT2ATSHR
SCHEMBL4670081 0.78 ADRB2 (0.42) ALDH1A1MAPK1ATMTSHRNPC1
SCHEMBL4673552 0.78 MAPK1 (0.49) ALDH1A1MAPK1ATMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054881-B1 NOVEL SULFONAMIDE SUBSTITUTED CHROMAN DERIVATIVES USEFUL AS BETA-3 ADRENORECEPTOR AGONISTS BAYER CORP (US) 2008-07-30 EP disclosed
US-6051586-A HYPOGLYCEMIC AGENTS; ANTIDIABETIC AGENTS BAYER CORPORATION (US) 2000-04-18 US disclosed