SCHEMBL4673352

SCHEMBL4673352

NC(=O)c1ccc(-n2nnn(CCCc3ccccc3)c2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.50
ATM Q13315 1/20 0.50
PLA2G10 O15496 1/20 0.42
PLA2G2A P14555 1/20 0.42
ROCK2 O75116 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CFTR P13569 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
PFKFB3 Q16875 1/20 0.39
TSHR P16473 2/20 0.39
OPRM1 P35372 2/20 0.39
OPRD1 P41143 2/20 0.39
PARP1 P09874 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
FAAH O00519 1/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4672123 0.85 MAPKAPK2 (0.46) ALDH1A1HPGDTSHRPARP1PARP2
SCHEMBL4673358 0.85 MAOB (0.46) ROCK2ALDH1A1PFKFB3TSHR
SCHEMBL4670084 0.85 ROCK2 (0.56) MAPK1ATMPLA2G10PLA2G2AROCK2
SCHEMBL4673552 0.80 MAPK1 (0.49) MAPK1ATMROCK2MEN1KMT2A
SCHEMBL4675102 0.79 ALDH1A1 (0.42) MAPK1ATMMEN1KMT2AALDH1A1
SCHEMBL4670479 0.79 ALDH1A1 (0.39) MAPK1ATMMEN1KMT2AALDH1A1
SCHEMBL4673671 0.78 SIGMAR1 (0.52) MEN1KMT2AALDH1A1
SCHEMBL4670081 0.77 ADRB2 (0.42) MAPK1ATMALDH1A1TSHROPRM1
Water SCHEMBL4673066 0.76 ADRB2 (0.41) MAPK1ATMALDH1A1TSHROPRM1
SCHEMBL4670624 0.76 PARP15 (0.40) MAPK1ATMALDH1A1TSHROPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054881-B1 NOVEL SULFONAMIDE SUBSTITUTED CHROMAN DERIVATIVES USEFUL AS BETA-3 ADRENORECEPTOR AGONISTS BAYER CORP (US) 2008-07-30 EP disclosed
US-6903218-B2 Sulfonamide substituted chroman derivatives BAYER PHARMACEUTICALS CORPORATION (US) 2005-06-07 US disclosed