SCHEMBL4672091

SCHEMBL4672091

Cn1nnn(-c2ccc(C(N)=O)cc2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43
ATM Q13315 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 2/20 0.42
BRD4 O60885 1/20 0.42
BRPF1 P55201 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
TSHR P16473 1/20 0.41
PTGS2 P35354 2/20 0.41
PABPC1 P11940 1/20 0.41
MAPKAPK2 P49137 1/20 0.40
ALPL P05186 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
ALPG P10696 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4675102 0.80 ALDH1A1 (0.42) ALDH1A1HPGDMAPK1ATMSMN1; SMN2
SCHEMBL2611112 0.75 PTGS2 (0.46) ALDH1A1SMN1; SMN2HSD17B10PTGS2POLB
SCHEMBL4670479 0.75 ALDH1A1 (0.39) ALDH1A1HPGDMAPK1ATMSMN1; SMN2
SCHEMBL8301872 0.74 ALDH1A1 (0.51) ALDH1A1HPGDMAPK1TSHRGAA
SCHEMBL4670084 0.72 ROCK2 (0.56) ALDH1A1HPGDMAPK1ATMMEN1
SCHEMBL4670468 0.71 PARP15 (0.42) ALDH1A1MAPK1ATMMEN1KMT2A
SCHEMBL4673352 0.71 MAPK1 (0.50) ALDH1A1HPGDMAPK1ATMMEN1
SCHEMBL4670421 0.71 PARP10 (0.42) ALDH1A1MAPK1ATMKDM4EMEN1
SCHEMBL2611117 0.71 GSK3A (0.47) ALDH1A1ATMKDM4EPTGS2GAA
SCHEMBL4673552 0.70 MAPK1 (0.49) ALDH1A1HPGDMAPK1ATMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054881-B1 NOVEL SULFONAMIDE SUBSTITUTED CHROMAN DERIVATIVES USEFUL AS BETA-3 ADRENORECEPTOR AGONISTS BAYER CORP (US) 2008-07-30 EP disclosed
US-6903218-B2 Sulfonamide substituted chroman derivatives BAYER PHARMACEUTICALS CORPORATION (US) 2005-06-07 US disclosed
US-6051586-A HYPOGLYCEMIC AGENTS; ANTIDIABETIC AGENTS BAYER CORPORATION (US) 2000-04-18 US disclosed