SCHEMBL467215

SCHEMBL467215

COc1ccc(CCl)cc1.[MgH2]

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.56
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA7 P43166 1/20 0.55
CA9 Q16790 1/20 0.55
CA14 Q9ULX7 1/20 0.55
AGXT P21549 2/20 0.52
LTA4H P09960 1/20 0.52
TAAR1 Q96RJ0 1/20 0.52
ALDH1A1 P00352 3/20 0.52
ALOX15 P16050 2/20 0.52
KDM4E B2RXH2 1/20 0.52
MAPT P10636 1/20 0.52
CMA1 P23946 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.50
TP53 P04637 1/20 0.50
CYP3A4 P08684 1/20 0.50
TSHR P16473 1/20 0.50
ALOX12 P18054 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13096 0.97 IDO1 (0.58) IDO1CA12CA1CA2CA7
SCHEMBL1657653 0.95 IDO1 (0.56) IDO1CA12CA1CA2CA7
SCHEMBL8993257 0.91 LTA4H (0.65) IDO1CA12CA1CA2CA7
SCHEMBL6157954 0.91 LTA4H (0.54) IDO1CA12CA1CA2CA7
SCHEMBL2996706 0.91 MAOB (0.59) IDO1CA12CA1CA2CA7
(Chloromethyl)Benzene SCHEMBL28005139 0.89 LTA4H (0.69) IDO1CA12CA1CA2CA7
SCHEMBL28148603 0.87 IDO1 (0.48) IDO1CA12CA1CA2CA7
SCHEMBL5505882 0.85 APP (0.67) IDO1AGXTALDH1A1MAPTSMN1; SMN2
SCHEMBL28784521 0.85 APP (0.67) IDO1AGXTALDH1A1MAPTSMN1; SMN2
Bicarbonate SCHEMBL28421098 0.83 CA1 (0.52) IDO1CA1CA2ALDH1A1CMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100548950-C Process for preparing esters and ethers of probucol and derivatives thereof ATHEROGENICS INC (US) 2009-10-14 CN claimed
CN-1759084-A Process for preparing esters and ethers of probucol and derivatives thereof ATHEROGENICS INC (US) 2006-04-12 CN claimed
US-20260042736-A1 COMPOSITIONS AND METHODS FOR MAKING SCYTONEMIN AND ITS ANALOGS AND DERIVATIVES Board of Regents of Nevada System of Higher Education on behalf of the University of Nevada Reno (US) 2026-02-12 US disclosed
CN-116102407-B Method for preparing gastrodia elata extract 2, 4-bis (4-hydroxybenzyl) phenol 北京化工大学 2024-07-23 CN disclosed
CN-116102407-A Method for preparing gastrodia elata extract 2, 4-bis (4-hydroxybenzyl) phenol 北京化工大学 2023-05-12 CN disclosed
CN-112047919-B Ticagrelor intermediate and preparation method thereof 常州制药厂有限公司 2021-06-18 CN disclosed
CN-112047919-A Ticagrelor intermediate and preparation method thereof 常州制药厂有限公司 2020-12-08 CN disclosed
EP-2399577-A1 Use of N-containing spirocompounds for the enhancement of cognitive function Adolor Corporation (US) 2011-12-28 EP disclosed
US-8022060-B2 Spirocyclic heterocyclic derivatives and methods of their use ADOLOR CORPORATION (US) 2011-09-20 US disclosed
US-20110218186-A1 SPIROCYCLIC HETEROCYCLIC DERIVATIVES AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2011-09-08 US disclosed
US-20100029614-A1 SPIROCYCLIC HETEROCYCLIC DERIVATIVES AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2010-02-04 US disclosed
US-7230139-B2 Diterpenoid compounds, compositions thereof and their use as anti-cancer or anti-fungal agents GEMIN X BIOTECHNOLOGIES (CA) 2007-06-12 US disclosed
US-7217844-B2 Diterpenoid compounds, compositions thereof and their use as anti-cancer or anti-fungal agents GEMIN X BIOTECHNOLOGIES (CA) 2007-05-15 US disclosed
US-20060270695-A1 Spirocyclic heterocyclic derivatives and methods of their use CUBIST PHARMACEUTICALS, INC. 2006-11-30 US disclosed
WO-2006105442-A2 SPIROCYCLIC HETEROCYCLIC DERIVATIVES AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2006-10-05 WO disclosed
CN-1759084-A Process for preparing esters and ethers of probucol and derivatives thereof ATHEROGENICS INC (US) 2006-04-12 CN disclosed
US-20050070540-A1 Diterpenoid compounds, compositions thereof and their use as anti-cancer or anti-fungal agents GEMIN X PHARMACEUTICALS CANADA INC. (CA) 2005-03-31 US disclosed
US-20050032802-A1 Diterpenoid compounds, compositions thereof and their use as anti-cancer or anti-fungal agents GEMIN X BIOTECHNOLOGIES INC. 2005-02-10 US disclosed
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed
US-5260451-A Enzyme inhibitors MERCKLE GMBH (DE) 1993-11-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110218186-A1 SPIROCYCLIC HETEROCYCLIC DERIVATIVES AND METHODS OF THEIR USE OPRK1, OPRD1, OPRL1 IDO1 1463/4885CA12 2102/4885CA1 1362/4885
US-20260042736-A1 COMPOSITIONS AND METHODS FOR MAKING SCYTONEMIN AND ITS ANALOGS AND DERIVATIVES TDO2, SCO2, TPH1 IDO1 8/4885CA12 2255/4885CA1 2967/4885
US-20050070540-A1 Diterpenoid compounds, compositions thereof and their use as anti-cancer or anti-fungal agents CYP51A1, ERG28, BAD IDO1 467/4885CA12 896/4885CA1 1596/4885
US-20100029614-A1 SPIROCYCLIC HETEROCYCLIC DERIVATIVES AND METHODS OF THEIR USE OPRK1, OPRD1, OPRL1 IDO1 1463/4885CA12 2102/4885CA1 1362/4885
US-20060270695-A1 Spirocyclic heterocyclic derivatives and methods of their use OPRK1, OPRD1, OPRL1 IDO1 1463/4885CA12 2102/4885CA1 1362/4885
US-20050032802-A1 Diterpenoid compounds, compositions thereof and their use as anti-cancer or anti-fungal agents CYP51A1, ERG28, BAD IDO1 467/4885CA12 896/4885CA1 1596/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.