SCHEMBL4673533

SCHEMBL4673533

O=c1n(CCCOc2ccc(F)cc2)nnn1-c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.44
MAPT P10636 3/20 0.44
GAA P10253 1/20 0.44
HSPB1 P04792 1/20 0.44
PKM P14618 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HRH3 Q9Y5N1 1/20 0.43
KMT2A Q03164 4/20 0.43
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
MEN1 O00255 3/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
POLB P06746 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PTGS1 P23219 2/20 0.40
LTA4H P09960 1/20 0.40
PTGS2 P35354 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6300285 0.84 NPC1 (0.41) HRH3DRD2DRD3POLB
SCHEMBL6300283 0.80 PARP10 (0.47) HRH3KMT2AMEN1
SCHEMBL4672086 0.77 KCNJ1 (0.53) MAPTGAASMN1; SMN2KMT2AMEN1
SCHEMBL4670082 0.76 KMT2A (0.48) MAPTPKMSMN1; SMN2KMT2AMEN1
SCHEMBL4670425 0.75 KMT2A (0.43) MAPTPKMSMN1; SMN2KMT2AMEN1
SCHEMBL28180201 0.75 HSPB1 (0.66) MAPTGAAHSPB1HRH3KMT2A
SCHEMBL28180988 0.75 HSPB1 (0.70) ENPP2MAPTGAAHSPB1HRH3
SCHEMBL4673671 0.74 SIGMAR1 (0.52) MAPTPKMSMN1; SMN2KMT2AMEN1
SCHEMBL4672275 0.73 ALDH1A1 (0.44) MAPTPKMSMN1; SMN2KMT2AMEN1
SCHEMBL4675267 0.72 ALDH1A1 (0.41) MAPTPKMSMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054881-B1 NOVEL SULFONAMIDE SUBSTITUTED CHROMAN DERIVATIVES USEFUL AS BETA-3 ADRENORECEPTOR AGONISTS BAYER CORP (US) 2008-07-30 EP disclosed